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(2S)-N-(dimethyl-1H-1,2,4-triazol-3-yl)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carboxamide
3-(1H-imidazol-4-ylmethyl)-4-[4-(piperidin-1-yl)butanoyl]piperazin-2-one
N-{[3-methyl-7-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}pyrazine-2-carboxamide
2-(4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-1-yl)pyridine-3-carboxamide
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-5-(methoxymethyl)thiophene-2-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-benzyl-2-[4-(4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[2-(pyridin-4-yl)ethyl]propanamide
2-{[(3,5-dimethoxyphenyl)methyl]amino}-N-(3-fluoro-2-methylphenyl)acetamide
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)acetamide
5-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
9-(2-hydroxyacetyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)pyridin-2-amine
(2R,3R,6R)-5-(1H-indole-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazole
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(3-hydroxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(4-oxo-4H-chromen-6-yl)piperazine-1-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-methyl-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}urea
1-({2-[({1,9-dioxaspiro[5.5]undecan-4-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]acetamide
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)but-3-en-1-one
N-methyl-2,6-dioxo-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinazolin-2-one
N-methyl-2-(methylsulfanyl)-N-(pyrazin-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-hydroxypyridine-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-hydroxy-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]piperidine-4-carboxylate
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-(6-chloro-2-methylpyridin-3-yl)-4-(4-methoxypyrimidin-2-yl)piperazine-1-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
3-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-6-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-1H-indole
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-{1-[(5-methylthiophen-2-yl)methyl]azepan-3-yl}pyrazolo[1,5-a]pyridine-3-carboxamide
1-cyclopropanecarbonyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidine-4-carboxamide
5-(oxolan-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}thiophene-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl]pyridine-2-carboxamide
7-[(2-fluorophenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(pentan-3-yl)acetamide
N-(5-fluoro-2-methylphenyl)-2-{[2-(methylamino)pyridin-4-yl]formamido}propanamide
(1S,5R)-3-(pyridine-3-carbonyl)-6-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
1-oxo-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
(1S,5R)-6-(cyclopropylmethyl)-N-(2,4-difluorophenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(1H-indole-6-carbonyl)pyrrolidine-2-carboxamide
ethyl({[2-(trifluoromethoxy)phenyl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine