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N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-ethyl-5-[7-fluoro-4-(thiomorpholine-4-carbonyl)quinolin-2-yl]pyrimidin-2-amine
N-[2-(4-chlorophenyl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-(methylamino)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyridine-3-carboxamide
4-[6-(5-fluoro-2-methylphenyl)pyridine-3-carbonyl]morpholine
ethyl 2-{1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}acetate
5-{4-hydroxy-1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(morpholin-4-yl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propan-1-one
4-{[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
ethyl 2-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}amino)acetate
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-(pyridin-4-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[3-cyclopropyl-5-({[(2-methylphenyl)methyl]sulfanyl}methyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(propan-2-ylsulfanyl)ethyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-[4-(furan-2-yl)phenyl]urea
(3S,4R)-3-benzyl-4-methyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-ol
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-[(3S,4R)-1-[(2,3-dichlorophenyl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-hydroxypiperidine-4-carboxylic acid
(1S,5S,6R,7R)-3-cyclohexyl-6-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-{2-[(dimethylamino)methyl]-4-(pyrazin-2-yl)phenoxy}-N-(2-methoxy-5-phenylphenyl)acetamide
(1S,5R)-3-(4-aminopyrimidin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylthiophene-2-carboxamide
N-cyclopropyl-3-{1-[3-(3,4-difluorophenyl)propanoyl]piperidin-3-yl}propanamide
1-[1'-(dimethyl-1,3-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
5-fluoro-2-(4-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}piperazin-1-yl)pyrimidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-methylthiophene-2-carboxamide
5-(5-fluoro-2-methylphenyl)pyridin-2-amine
5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
(1S,4S)-2-(3,4-difluorophenyl)-5-[3-(1H-indol-3-yl)propanoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(thiophen-2-yl)propanamide
1-[2-(dimethylamino)-4-({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
2-(methoxymethyl)-1-[(5-phenylthiophen-2-yl)methyl]piperidine
(4aR,7aS)-N,N-dimethyl-4-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(5-{1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
1-[4-(4-methylphenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxamide
7-(4-chloro-2-hydroxybenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(2-methoxyphenoxymethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-3-carboxamide
1-methyl-9-[(2,4,6-trimethylphenyl)methyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-(1-benzylpiperidin-3-yl)-4-(3-chlorophenyl)piperazine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
1-(3-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
2-[2-(4H-1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one