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N'-(2,4-dimethylphenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}ethanediamide
N-{3-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropyl}-3-methoxybenzamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(2-fluorophenyl)methyl]-N-methylpiperidin-3-amine
N-(1-methyl-1H-pyrazol-4-yl)-4-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)benzamide
4-chloro-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-methoxybenzamide
2-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2-azaspiro[4.4]nonan-3-one
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrazol-1-yl)acetamide
2-[4-(2-ethylbutyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-methoxy-N-[2-(pyridin-3-yloxy)propyl]-5-sulfamoylbenzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-propyl-1,3-thiazole-4-carboxamide
3-[4-(4-methanesulfonylphenyl)-1H-pyrazol-1-yl]propanamide
1-(4-{4-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]piperazin-1-yl}phenyl)ethan-1-one
6-[(3-chloro-4-hydroxyphenyl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-benzyl-5-(furan-3-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
(1S,5R)-3-(1-benzoylpiperidin-4-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
(3R,4R)-7-(pyrimidin-5-yl)-3-(pyrrolidin-1-yl)-3,4-dihydro-2H-1-benzopyran-4-ol
6-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(4aS,7aR)-4-[2-(dimethylamino)acetyl]-N,N-diethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
7-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-methyl-5-({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrrolidin-2-one
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
methyl 4-{4-oxo-7-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}benzoate
2-(4-{[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]methyl}phenoxy)acetic acid
N-(1-carbamoylcyclopentyl)-2-(ethylamino)pyrimidine-5-carboxamide
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]acetamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
2,3,5-trimethyl-6-{[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrazine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-(5-methyl-1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
5-chloro-4-{1-cyclohexyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-dimethyl-1H-pyrazole
N6-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
methyl (1R,3S,3aR,6aS)-1,5-diethyl-3-(4-ethynylphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N4-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)morpholine-2-carboxamide
[(3R,4R)-1-(3-fluoropyridine-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[2-(pyridin-3-yl)ethyl]pyrrolidin-2-one
1-(1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclopentyl)pyrrolidine
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
8-methoxy-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3aS,6aR)-5-benzoyl-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
1-[(4-fluorophenyl)methyl]-4-(2-methyl-1,3-thiazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
1-{2-oxo-2-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyridin-2-one
(2S,4R)-4-(dimethylamino)-1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)pyrrolidine-2-carboxylic acid
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-3-(2-oxoimidazolidin-1-yl)benzamide