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4-{1-[2-(dimethylamino)acetyl]piperidin-3-yl}benzoic acid
(1R,5R)-N-(3-fluorophenyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(3-methylphenyl)piperidin-1-yl]propan-1-one
2-{5-[(carbamoylamino)methyl]-1-(2,5-dichlorophenyl)-1H-1,2,4-triazol-3-yl}acetamide
N-(2-hydroxyethyl)-2-(2-hydroxyphenoxy)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(propan-2-ylsulfanyl)acetamide
2-methyl-N-{2-[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
(3S,4S)-1-(6-chloro-2-methylquinoline-4-carbonyl)-4-methylpiperidine-3,4-diol
4-[(4-methoxyphenyl)methyl]-1-(1-methylcyclohexanecarbonyl)-1,4-diazepan-5-one
1-ethyl-4-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}-1H-pyrrole-2-carbonitrile
3-{2-[2-(3-chlorophenyl)-1H-imidazol-1-yl]ethyl}pyridine
1-(3-fluorophenyl)-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethan-1-ol
7-(5-chloropyridin-2-yl)-4-[(4-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}azepane-2-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}propanamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[4-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)quinoline-2-carboxamide
5-cyclopropanecarbonyl-3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N7-(3-methoxyphenyl)-2,N3,N3-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3,7-dicarboxamide
3-{[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-4H-chromen-4-one
N-[1-(dimethylamino)butan-2-yl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-{2-[3-(3-methylphenoxy)azetidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-amino-4-(3-hydroxyphenyl)-6-(2,4,5-trifluorophenyl)pyridine-3-carbonitrile
N-[(2,4-dichloro-6-methylphenyl)methyl]morpholine-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-hydroxy-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(2-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
4-methyl-3-[({2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}carbamoyl)amino]benzamide
N-(2-methoxyphenyl)-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
5-{[3-(dimethylamino)-2,2-dimethylpropyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-4-carbonitrile
2-(butylsulfanyl)-N4-methyl-N4-(pyrazin-2-ylmethyl)pyrimidine-4,6-diamine
4-(5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-8-methyl-3,4-dihydroquinazolin-4-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]propanamide
2-(adamantan-1-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1-[4-(propylsulfamoyl)phenyl]urea
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(2-methylphenoxy)piperidine
5,8-dimethyl-2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-fluoro-2-methoxybenzamide
N,2,6-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}quinoline-4-carboxamide
1-(3-chlorophenyl)-4-(4-fluorobutyl)piperazin-2-one
2-cyclopentyl-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(2-{[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-{2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
(3-{[1-(oxane-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[4-(methylsulfanyl)phenyl]acetamide
2-cyclopentyl-9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-fluorobenzene-1-sulfonamide