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3-(2-methoxyphenyl)-6-[3-(1H-pyrazol-5-yl)phenyl]pyridazine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[(3S)-pyrrolidin-3-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-(2-fluorophenoxymethyl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1H-pyrazole-3-carboxamide
1-(2,3-dihydro-1H-inden-5-yl)-3-(oxan-4-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(naphthalen-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
7-(cyclopropylmethyl)-2-(5-phenyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{[2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[3-(propan-2-yl)phenyl]-4-{[(pyridin-3-yl)carbamoyl]methyl}piperazine-1-carboxamide
1-({4-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-3-methoxyphenyl}methyl)piperidine-4-carbonitrile
N,3,4,7-tetramethyl-N-[(3-methylpyridin-4-yl)methyl]-1H-indole-2-carboxamide
4-cyclopropyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
4-ethyl-5-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methyl-1,3-thiazole
9-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.6]dodecane
2-(2-chloro-4-fluorophenyl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}pyrimidin-2-yl)morpholine
2-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-benzofuran-7-carboxamide
N-{4-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
N-(3-fluoro-4-methylphenyl)-2-{4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]morpholin-3-yl}acetamide
2-[ethyl(2-methoxyethyl)amino]-2-(5-fluoro-2-methoxyphenyl)acetic acid
N-(4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenyl)acetamide
2-methanesulfonamido-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
(3aS,6aS)-2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(6-ethyl-2-methylquinoline-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 2-(2-fluoro-5-methoxyphenyl)pyridine-3-carboxylate
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
N,N-dimethyl-3-[2-(2-methylphenyl)ethyl]piperidine-1-sulfonamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(pyridin-3-yl)ethyl]piperidin-2-one
6-(4-fluoro-3-methylbenzoyl)-2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(pyridin-2-ylmethyl)amine
1-(4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carbonyl)piperidine-3-carboxamide
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenoxyethan-1-one
methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]but-3-enamide
methyl 5-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
5-ethyl-1'-(3,4,5-trifluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
4-butyl-11-[(2-methylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 5-{[(3,4-difluorophenyl)methyl]amino}-1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-cyclohexyl-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazin-2-yl)ethan-1-ol
2-[(4aR,7aS)-4-(cyclopentylcarbamoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-[1-(cyclohexylmethyl)-4-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
1-(2,6-difluoro-4-methoxybenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-(4-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}phenoxy)pyrimidine
(3S,4S)-3-hydroxy-4-[(7-methoxy-3,7-dimethyloctyl)(methyl)amino]-1λ6-thiolane-1,1-dione