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1-{2-[4-(2-phenylethyl)piperazin-1-yl]pyrimidin-4-yl}piperidin-3-ol
N-tert-butyl-2-(1-methyl-1H-imidazol-2-yl)-N-(pyridin-2-ylmethyl)benzamide
1-[3-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-2-methoxyethan-1-one
3-[methyl({2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl})amino]-1λ6-thiolane-1,1-dione
2,4-dimethoxy-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
2-[methyl(piperidin-4-yl)amino]-N-[(4-phenylphenyl)methyl]acetamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
N-[(5-ethylpyridin-2-yl)methyl]-3-fluoro-N,8-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N-methyl-5-phenoxy-N-[1-(pyridin-3-yl)ethyl]furan-2-carboxamide
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
3-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-(propan-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-2-one
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-3-(1H-imidazol-2-yl)piperidine
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
6-methyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N,1-dimethyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-methylpiperazin-1-yl)propyl]benzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(4-fluorophenyl)methyl]-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-[({2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}amino)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
(2R)-2-[5-(3-methyl-1,2-benzoxazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-(4-chloro-3-methoxyphenyl)-2-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}acetamide
2-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)benzonitrile
4-(3-chloro-5-fluorophenyl)-7-hydroxy-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
1-(furan-2-ylmethyl)-4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}piperidine
N-[(2-chlorophenyl)methyl]-1-ethyl-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N-[2-(pyrazin-2-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(1-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
5-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
(2S,4R)-4-amino-N-ethyl-1-[4-(4-hydroxyphenyl)benzoyl]pyrrolidine-2-carboxamide
(1S,5R)-6-benzyl-3-(5-phenyl-1,2,4-oxadiazol-3-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(thiophen-2-ylmethyl)propanamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(2,3-difluoro-6-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N,N-dimethylpyridine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-cyclohexyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methylpropanamide
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
N,1,3-trimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-({3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
[4-(2,3-dihydro-1-benzofuran-5-yl)pyridin-2-yl]methanol
2-(furan-2-yl)-5-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidine
3,5-dichloro-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylbenzamide
2-(4-methoxyphenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-(4-chlorophenyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-ethyl-8-{[3-(2-methylphenyl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(diethylamino)ethyl]-N-ethyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide