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3-(3-methoxyphenyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
3-(azocan-1-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
2-{4-[4-(azepane-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
N-cyclopropyl-1-[1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-cyclopropyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethylpyrimidine-5-carboxamide
(1R,2R,6S,7S)-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-5-methylphenol
N-(2-methoxyethyl)-N,5-dimethyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1H-pyrrole-2-carboxamide
ethyl 4-({4-[(4-methylphenyl)methyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}amino)piperidine-1-carboxylate
1-{4-chloro-3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
5-[(4-ethylpiperazin-1-yl)methyl]-N-(5-methylhexan-2-yl)-1,2-oxazole-3-carboxamide
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
3-[(3R,4S)-1-(2-methyl-1H-pyrrole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(pyridin-3-yl)propan-1-one
3-(2-ethylbutyl)-8-[2-(morpholin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(4-{4-[(adamantan-2-yl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
1,3-dimethyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(2-hydroxypropanoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S)-4-methanesulfonyl-2-[(3,4,7-trimethyl-1H-indol-2-yl)formamido]butanoic acid
1-[2-(cyclohex-1-en-1-yl)ethyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
(1S,5R)-3-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
methyl 8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(cyclohexylmethyl)-5-[(furan-2-ylmethyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-(2-hydroxyethyl)-3-(1,3-thiazol-2-ylmethyl)urea
1-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
5-cyclopropyl-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1,3,4-oxadiazol-2-amine
[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
9-(cyclopropylmethyl)-1-methyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butan-1-ol
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide
propyl 4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
2-amino-N-(cyclohex-1-en-1-ylmethyl)-6-methylpyrimidine-4-carboxamide
2-(phenylsulfanyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
2-amino-6-(2,3-dimethylphenyl)-4-(pyridin-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidin-2-one
4-[(6-ethyl-2-methylpyrimidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methylpentan-1-one
3-(3-methoxyphenyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
5-(4-methylphenyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
dimethyl({2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(5-methylfuran-2-yl)ethyl})amine
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-methoxypiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-butyl-1-methyl-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
6-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-methyl-1-{2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(furan-2-ylmethyl)-5-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine