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3-[5-(dimethyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amine
3-({methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)phenol
4-{1-[6-(1,2,3,6-tetrahydropyridin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
N-(2-hydroxyethyl)-4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-2-carboxamide
3-fluoro-4-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
1-cyclopentanecarbonyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
N-[2-(4-{3,9-diazaspiro[5.5]undecane-3-carbonyl}phenoxy)ethyl]acetamide
(1s,4s)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-hydroxycyclohexane-1-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]propanamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyrrolidine-3-carboxamide
3-(2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}acetamido)propanoic acid
(3S,4R)-1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-methylpiperidine-3,4-diol
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-6-phenylpyridine-3-carboxylic acid
3-methoxy-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
6,7-dimethoxy-2-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(3-{2-[1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-(2-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-(3-methylpyridin-4-yl)-4-(2,4,5-trifluorobenzoyl)-1,4-diazepane
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-methyl-N-[(4-phenoxyphenyl)methyl]oxolane-3-carboxamide
1-cyclohexyl-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-3-(2-methoxyethyl)-1H-1,2,4-triazole
N-(1-cyanocyclopentyl)-2-(2,3-dihydro-1H-inden-1-yl)acetamide
(3R,4R)-4-cyclopropyl-4-hydroxy-3-methyl-N-(2-phenylethyl)piperidine-1-carboxamide
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)benzamide
3-(propan-2-yl)-5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(2-acetylphenyl)-3-[2-(2-hydroxyethyl)piperidin-1-yl]propanamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-{1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-[2-(propan-2-yloxy)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
[3-ethyl-1-(2-methoxy-4-methylbenzoyl)piperidin-3-yl]methanol
1-(2,2-diphenylethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
[(3R,4R)-1-(dimethyl-1,3-thiazol-2-yl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(2S,4S)-4-[2-(3-chloro-2,6-difluorophenyl)acetamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-ethyl-N-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
(1S,5R)-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[2-(difluoromethoxy)phenyl]methyl}-1,4-oxazepan-5-one
3-[2-(trifluoromethyl)morpholine-4-carbonyl]benzene-1,2-diol
ethyl 4-[6-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(thiophene-2-carbonyl)piperidine
2-amino-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-4-carboxamide