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[(3S,5R)-1-(5-chlorothiophene-2-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
2-methoxy-1-(1'-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
2-methyl-N-{2-oxo-2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}propanamide
4-hydroxy-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-phenylpyrimidine-5-carboxamide
3-(3-methoxyphenoxy)-1-[(5-propylfuran-2-yl)methyl]azetidine
(3R,4R)-4-amino-1-({2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)piperidin-3-ol
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-(4-methoxyphenyl)furan-2-carboxamide
3-(1H-imidazol-4-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-ethyl-1-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)urea
N'-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N'-(2-methoxyethyl)-N,N-dimethylbutanediamide
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-(oxan-4-yl)acetamide
3-(2-hydroxy-1-phenylethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-(4-methoxy-2-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenyl)-1H-pyrazole
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methoxyphenoxy)acetamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{[3-oxo-3-(pyrrolidin-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(2-amino-9H-purin-6-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N,N-dimethyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[3-(cyclopropylmethyl)-1-(2-methoxy-6-methylbenzoyl)piperidin-3-yl]methanol
1'-benzyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,3'-piperidine]-6'-one
4-{4-[1-(1,2,2,6,6-pentamethylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]phenyl}but-3-yn-1-ol
4-({4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)pyridine
(2S,4S)-N,N-diethyl-4-(3-hydroxybenzamido)-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1H-pyrazole-4-carboxamide
5-(1H-imidazol-2-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazole
1-(3-phenylphenyl)-N-(piperidin-3-yl)piperidin-4-amine
ethyl 2-[({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)(methyl)amino]acetate
N-[2-(dimethylamino)ethyl]-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}furan-3-carboxamide
5-[({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)methyl]-N-methylfuran-2-carboxamide
2-[(dimethylamino)methyl]-4-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenol
1-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-methylpentane-1,2-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(1H-imidazol-1-yl)-N-(pentan-3-yl)acetamide
3-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
2-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-(methylamino)pyridine-3-carboxamide
2-(4-chlorophenyl)-4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]morpholine
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethylamino)ethyl]-3-phenylpropanamide
4-(1H-imidazol-2-yl)-3-(4-methoxyphenyl)-1H-pyrazole
9-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]-3,9-diazaspiro[5.5]undecane-2,4-dione
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-(2-methoxyethoxy)ethan-1-one
2-(morpholin-4-yl)-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-cyclopropyl-6-oxo-N-(pentan-3-yl)piperidine-3-carboxamide
(4aR,7aS)-1-acetyl-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-fluoro-4-methylbenzenesulfonyl)-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one