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1-(4-phenyl-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-yl)ethan-1-one
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
1-[4-(methylamino)pyrimidin-2-yl]-4-(pyrrolidine-1-carbonyl)-1,4-diazepan-6-ol
5-[3-(morpholin-4-ylmethyl)phenyl]furan-2-carboxylic acid
2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-1,3-benzodiazole
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(3-hydroxy-6-methylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyridine-3-carboxamide
1-(3-chloro-4-methoxyphenyl)-4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}pyrrolidin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
3-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-4-methoxybenzoic acid
N-cyclohexyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-methylphenyl)methyl]acetamide
2-{4-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-2-(methylamino)acetamide
1-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
1-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(furan-2-ylmethyl)-4-(3-phenylpiperazin-1-yl)pyridine-2-carboxamide
2-methoxy-5-{1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-(4-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}phenyl)-2-methylbutan-2-ol
ethyl 1-({3-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carboxylate
14-(2-butoxy-3-methoxyphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-(3,4,5-trimethoxyphenyl)acetamide
4-[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-5-methylpyrimidin-2-amine
2-{4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]morpholin-3-yl}acetic acid
N-{2-[2-methyl-2-(pyrrolidin-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]-3-(pyridin-4-yl)propanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[(3-fluorophenyl)methyl]-6-methyl-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(4S)-1-[(3,5-dichloropyridin-4-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
3-(5-methylthiophen-2-yl)-5-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
(3R,4R)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
4-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2,6-dimethoxyphenol
N-benzyl{[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]amino}sulfonamide
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-9H-purin-2-amine
(1R,5S,6R)-N-methyl-3-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
N,N,5-trimethyl-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)oxane-4-carboxamide
2-ethyl-1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}butan-1-one
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
3-(1H-1,3-benzodiazol-2-yl)-1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]propan-1-one
N'-(3-ethylphenyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]butanediamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
1-[(2-aminopyridin-3-yl)methyl]-4-(furan-2-carbonyl)-1,4-diazepan-6-ol
1-(2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl](methyl)amino}ethyl)piperidin-2-one