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N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(1S,5R)-3-benzyl-6-(2,4-dimethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
4-[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-thiazole
methyl (2S)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxylate
5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-4-carboxamide
5-methoxy-2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-3-yl)acetamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-4-yl)ethyl]propanamide
5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-ethyl-3-({[3-(4-methylpiperazin-1-yl)butyl]carbamoyl}amino)benzamide
2-amino-N,3-diethyl-N-[2-(phenylsulfanyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3aR,5R,6S,7aS)-2-(2-methyl-6-propylpyrimidin-4-yl)-octahydro-1H-isoindole-5,6-diol
5-(adamantan-1-ylmethyl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
3-benzoyl-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
[1-({1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-[(2-ethyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-(quinolin-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-(difluoromethyl)-2-[4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-[1-(furan-2-carbonyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
(4aS,7aR)-1-(2,3-dimethoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,3R)-3-(4-phenyl-1H-1,2,3-triazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(3-methyl-4-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl)acetic acid
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
N-[2-(4-chlorophenyl)ethyl]-N-(pyridin-3-ylmethyl)morpholine-2-carboxamide
(3S,4R)-1-(oxane-4-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(3S,4S)-4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-1-cyclopentylpyrrolidin-3-ol
2-(3-acetyl-1H-pyrazol-1-yl)-N-(1-ethyl-1H-indazol-3-yl)acetamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-3-yl}propan-1-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(2-oxoazonan-1-yl)acetamide
3-(1H-1,3-benzodiazol-1-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
5-methyl-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
7-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
6-{3-[1-(dimethylamino)ethyl]phenyl}pyridine-3-carboxamide
3-fluoro-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(4-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperazine-1-carboxamide
5-chloro-3-methyl-N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}-1H-indole-2-carboxamide