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1-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]cyclopentane-1-carboxamide
2-(morpholin-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
N-[3-(3-chlorophenyl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
1-methyl-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-(2-methoxyethyl)-1-methyl-4-(pyridin-3-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperazine-1-carbaldehyde
N-[2-(diethylamino)ethyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
5,6-dimethyl-3-(quinolin-5-yl)-1,2-dihydropyridin-2-one
1-phenylmethanesulfonyl-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{[1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-6-oxo-1-propylpiperidine-3-carboxamide
2-[1-(cyclohexylmethyl)-4-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
(8aS)-2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[2-(2,3-dichlorophenyl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-({5-[(4-acetylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
9-[2-(4-fluorophenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-{1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
methyl 4-[(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N1,5-bis(2-methylpropyl)piperidine-3,5-dicarboxamide
2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-6-methylpyridin-3-ol
4-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrimidin-2-amine
(3S,4S)-1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-[1-(pyridin-4-yl)propyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(pyridin-2-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{1-[4-(furan-2-yl)phenyl]piperidin-4-yl}-N-methylpiperidin-4-amine
7-(5-tert-butyl-2-methoxybenzenesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-3-benzoyl-6-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-hydroxy-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-phenylpyrimidine-5-carboxamide
5-fluoro-2-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
6-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(2,4-dimethylbenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N,4-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
1-{[(2R,5S)-5-[(6-methoxypyridin-3-yl)methyl]oxolan-2-yl]methyl}piperidine-4-carboxylic acid
methyl 6-(2-phenylpropanoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-methyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]pyridin-2-amine
3-(1-hydroxy-3-methylbutan-2-yl)-5-methyl-3,4-dihydroquinazolin-4-one
7-(5-methylthiophen-2-yl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 1-[2-hydroxy-3-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
(3S,4S)-4-(morpholin-4-yl)-1-[(3-phenoxyphenyl)methyl]pyrrolidin-3-ol
2-(3-chloro-5-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
N-[2-(4-methoxyphenyl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-(6-methylpyridine-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-fluorophenoxymethyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
6-(4-chlorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-3-ol
(3R,9R)-11-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
6-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]pyridin-3-ol
N-ethyl-5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrimidin-2-amine