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2-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]pyridin-3-ol
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(2R,3R,6R)-3-(4-methylphenyl)-5-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,7aR)-1-[(2-methylpyrimidin-5-yl)methyl]-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,2,6-trimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-4-carboxamide
N-(2-cyclopropylphenyl)-4-(2-phenoxyethyl)piperazine-1-carboxamide
2-amino-4-phenyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrimidine-5-carboxamide
methyl 2-{1-[(2-aminopyrimidin-5-yl)methyl]-3-oxopiperazin-2-yl}acetate
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
ethyl 5-benzoyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(furan-2-yl)propyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(4-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}phenyl)methanamine
1-ethyl-9-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(4-methoxy-2-methylphenyl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
[(3aS,6aS)-2-[6-(methoxymethyl)pyrimidin-4-yl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
8-(1-methyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,5-dimethyladamantane-1-carboxamide
N-{[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-methyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,9S)-11-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
methyl 2-(1-{[(3-fluorophenyl)carbamoyl]carbonyl}-3-oxopiperazin-2-yl)acetate
2,3-dimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,7aS)-1-[2-(thiomorpholin-4-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
3-benzyl-1-(3-methoxypropyl)-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-[2-(phenylsulfanyl)ethyl]-N3-(prop-2-en-1-yl)piperidine-1,3-dicarboxamide
3-[methyl({2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl})amino]-1-phenylpropan-1-ol
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-5-(methoxymethyl)thiophene-2-carboxamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
2-[(1S,5R)-3-[(3-chloro-2-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[2-methyl-1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
2-{3-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenoxy}ethan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylbenzamide
2-(2-methoxyethyl)-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-yl)-2-oxa-7-azaspiro[4.5]decane-7-carboxamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1,4-diazepan-6-ol
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-phenyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N-tert-butyl-4-(6-methoxypyridazin-3-yl)benzene-1-sulfonamide
N-[(3-methyloxetan-3-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)benzene-1-sulfonamide
2-(3,4-dichlorophenyl)-4-{thieno[2,3-d]pyrimidin-4-yl}morpholine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-methylpyridine-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(2-methanesulfonylethyl)-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazine
(3S,4S)-1-(4-carbamoyl-1,3-thiazol-2-yl)-4-propylpyrrolidine-3-carboxylic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-methylpiperidine