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(1R,5S,6R)-3-[(3-chloro-4-methoxyphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
5-(3-methylbutyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(cyclopropylmethyl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
N4-[4-(pyridin-2-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(methoxymethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]cyclobutane-1-carboxamide
methyl 1-benzyl-5-[(cyclohexylmethyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)oxy]pyridine
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(pyrimidin-4-yl)ethyl]acetamide
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(3-ethoxyphenyl)methyl]amino}ethan-1-ol
2-(3-phenyl-1,2,4-oxadiazol-5-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-{[(2,5-difluorophenyl)carbamoyl]methyl}acetamide
(2R,6S)-4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
3-methyl-5-(2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-fluorophenyl)methyl]-4-[2-(1H-imidazol-1-yl)ethyl]-2-(propan-2-yl)-1,4-diazepane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}oxolane-3-carboxamide
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
1-benzyl-5-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3,3-dimethyl-1-[(5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
(3S,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
3-cyano-5-fluoro-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
3-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetamido}-2-methyl-N-(1,3-thiazol-2-yl)benzamide
(3R,4S)-3,4-dimethyl-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
9-(2-hydroxybutanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1'-(5-ethyl-1,3,4-oxadiazol-2-yl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-[6-(3-fluorophenyl)pyridine-3-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}pyridine
1-(3-fluoropyridine-4-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
2-chloro-5-acetamido-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]benzamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidine
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-1H-1,2,3-benzotriazole-5-carboxamide
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
methyl 1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
4-[3-methyl-6-oxo-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylic acid
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-[(3-methylphenyl)methyl]piperazine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
1,1,1-trifluoro-2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}propan-2-ol
2-(propan-2-yl)-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
3-chloro-6-[4-(2-ethoxy-2-oxoethyl)piperazin-1-yl]pyridine-2-carboxylic acid
1-ethyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-1,2,4-triazole
N-methyl-1-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
1-methyl-3-propyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(2-phenoxyethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{6-[2-(4-fluorophenyl)morpholin-4-yl]pyrimidin-4-yl}piperidin-4-ol
[(2-fluoro-4,5-dimethoxyphenyl)methyl](isoquinolin-5-ylmethyl)methylamine
(3aS,6aS)-2-(phenylcarbamoyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid