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5-[(diethyl-1H-1,2,4-triazol-1-yl)methyl]-3-(thiophen-2-yl)-1,2,4-oxadiazole
4-[(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)methyl]benzoic acid
2-methyl-1-{3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
5-fluoro-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-methylbenzene-1-sulfonamide
2-[({1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
1-[(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidine-2-carbonyl]piperidine
2-(4-fluorophenyl)-4-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
methyl 4-[2-amino-3-cyano-6-(2,2-dimethyloxan-4-yl)-5-methylpyridin-4-yl]-1H-pyrazole-3-carboxylate
ethyl 2-[({1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]acetate
2-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-6-methoxyphenol
2-{5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}pyridine
1-acetyl-N-methyl-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
3-{[butyl(methyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-methyl-6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-2,3-dihydropyridazin-3-one
ethyl 4-(oxan-2-ylmethyl)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylate
2-(furan-2-yl)-5-{imidazo[1,2-a]pyridin-6-yl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(2-hydroxypropyl)-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(4-ethylpiperazin-1-yl)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
4-{5-[1-(1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}-1,4-oxazepane
6-ethyl-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-methylquinoline-4-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
[(2S,4R)-4-(dimethylamino)-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidin-2-yl]methanol
N,4-dimethyl-3-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)benzamide
7-(1,3-benzothiazol-2-yl)-4-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[4-(propylsulfamoyl)phenyl]urea
2-[ethyl(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]ethan-1-ol
1-{4-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
(1R,2S,6R,7S)-4-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
dimethyl({[4-methyl-5-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
(3S,4S)-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-(methoxymethyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-4-phenyl-9-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,9-diazaspiro[5.5]undecane
4-[(2,3-difluorophenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
5-(2,3-dihydro-1,4-benzodioxin-2-yl)-3-[(3,4-dimethoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazole
4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxan-4-yl)acetamide
2,6-dimethoxy-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyridine-3-carboxamide
6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1-methyl-1H-indole
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(3-methylpyridin-4-yl)methyl]propanamide
3-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]phenyl}propanoic acid
2-{[6-(7-methyl-1H-indol-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
(3R,4R)-1-(1H-imidazol-4-ylmethyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
6-(2H-1,3-benzodioxol-5-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide