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N-{[7-(3,4-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
1-[3-(1H-pyrazol-4-yl)benzoyl]-3-(thiophene-2-carbonyl)piperidine
2-{[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-cyclopropyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-[(2-chloro-5-fluorophenyl)methyl]-1,4-oxazepan-5-one
(1S,6R)-N-(4-acetylphenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
6-(2-methylpropyl)-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyrimidin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2-(4-methyl-1,4-diazepan-1-yl)acetic acid
[2-({4-[(2-aminopyridin-3-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
(4aR,7aS)-1-methanesulfonyl-4-(6-methylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-({[(3R,4R)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-1-(3,5-dimethylphenyl)piperazin-2-one
N-{2-[(1-tert-butyl-5-oxopyrrolidin-3-yl)formamido]ethyl}-4-fluorobenzamide
methyl 3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(3-methylpyridin-2-yl)methyl]pyridin-2-amine
(2S,4R)-4-amino-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
8-[(4-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}phenyl)imidazolidine-2,4-dione
N-[3-(4-methoxyphenyl)propyl]-6-(6-methoxypyridin-3-yl)pyridine-3-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1H-pyrazole-3-carboxamide
N-{[1-(thiophene-3-sulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
3-({1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)benzonitrile
2-(dimethylamino)-N-methyl-N-(2-phenyl-1-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl)acetamide
N-[(4-methoxypyridin-2-yl)methyl]-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
7-cyclopentyl-2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-benzyl-3-(3,5-difluoropyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
7-(1-benzothiophen-3-yl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methoxy-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyridine-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
benzyl(ethyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2-{2-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]phenoxy}propanamide
N-{[4-(furan-2-ylmethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
2-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]pyridine
5-(4-ethoxyphenyl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
4-cyano-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
(2S,4S)-4-(4-{2-[(2-chloropyridin-4-yl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
1-[6-chloro-3-(morpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]azocane
1-(2-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)azepan-2-one
2-(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-cyclopentyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-phenylacetamide
1-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide