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(1S,5R)-3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
methyl (2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
1-[2-(methylamino)pyrimidine-5-carbonyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-(3-cyano-4-ethoxyphenyl)-1-methyl-1-[1-(pyridin-3-yl)propyl]urea
[5-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)furan-2-yl]methanol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
3-{1-[6-(diethylamino)pyridin-3-yl]-1H-imidazol-2-yl}phenol
N-[3-(methylsulfanyl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
9-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
(4aS,8aR)-6-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
6-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
N-[(2-chlorophenyl)methyl]-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}propanamide
N-(2-methoxyethyl)-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-methoxy-N-(propan-2-yl)-N-{[1-(pyridin-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
8-(3,7-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxylic acid
1-(2-methylpropyl)-4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
8-(2,4-difluorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-chloro-6-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]pyridine-2-carboxylic acid
3-(4-methoxyphenyl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-cyclohexyl-4-(3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazin-2-one
1-(3-hydroxypyridine-2-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
3-(4-chlorophenyl)-5-(2,2-dimethyloxane-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3S,4S)-1-(1-cyclopropanecarbonylpiperidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-tert-butyl-2-(4-{[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}phenoxy)acetamide
[(3R,4R)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(4-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)-4-methoxypyrimidine
N-[5-(4-benzylpiperazine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]thiophene-2-carboxamide
N-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
11-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(furan-2-ylmethyl)-2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
(3S,4S)-4-propyl-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S)-3-phenyl-2-{[4-(piperidin-1-ylmethyl)phenyl]formamido}propanoic acid
1-(4-fluorophenyl)-4-(5-methoxypyrimidin-2-yl)-1,4-diazepane
[2,4,6-trimethyl-3-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)phenyl]methanol
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-3-methylthiophene-2-carboxamide
[(3R,4S)-1-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
8-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-[(4-fluorophenyl)methyl]-1,3-dimethyl-N-(2-methylpropyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(methylsulfanyl)-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propan-1-one
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide