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1-(cyclopropylmethyl)-5-(2,5-dimethoxybenzoyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-amine
(2R,6R)-4-(2-fluorobenzoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[(2-chlorophenyl)methyl]propanamide
methyl 6-[(2-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[3-(morpholin-4-yl)propyl]-4-(piperidin-3-yl)benzamide
(2S)-3-phenyl-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}propanoic acid
4-{[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}benzene-1,3-diol
3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-6-methoxyquinolin-2-ol
2-methoxy-1-{1'-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-methyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrrole-3-carbonitrile
2-(2,4-difluorophenoxy)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-2,5-dimethyl-N-(thiophen-3-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(2-methoxyphenoxy)-N-{[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}acetamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(thiophen-2-yl)butan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-cyclohexyl-N-methyl-1H-pyrazole-4-carboxamide
1-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)butan-2-ol
1-[3-(cyclopentyloxy)phenyl]-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
3-{1-[2-(4-methoxyphenoxy)ethyl]pyrrolidin-2-yl}-5-(propan-2-yl)-1,2-oxazole
7-(4-chlorophenyl)-2-(1,3-thiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinoline
2-(dimethylamino)-N-[(3R,4S)-4-propyl-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
5-(methoxymethyl)-3-methyl-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazole
6-methyl-2-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-4-carboxamide
4-[2-(1H-imidazol-1-ylmethyl)pyrrolidin-1-yl]-6-methoxypyrimidin-2-amine
3-(azocane-1-carbonyl)-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-ethylpropanamide
2-amino-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
9-(2-methoxyethyl)-4-[(4-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)quinolin-6-yl]acetamide
N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N3-(cyclohexylmethyl)-N5-(2,3-dihydro-1H-inden-2-yl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
(1R,5R)-N,N-dimethyl-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-ethyl-4,4,4-trifluoro-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)butanamide
(1R,9S)-5-amino-12-methyl-3-(1-methyl-1H-pyrazol-4-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
6-(3-fluoro-5-methylphenyl)-2-methyl-[1,2,4]triazolo[1,5-a]pyridine
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-(3-hydroxypropyl)-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(3-methoxypropyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
5-{[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]methyl}-N,N-dimethylpyridin-2-amine
2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}acetamide