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(3aS,6aR)-5-[(4-fluoro-2-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{2-[(4-butylpiperazin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyrimidin-4-amine
4-[4-(naphthalen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-{2-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
1-cyclohexyl-4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1H-pyrrole-2-carbonyl)piperazine
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-2,1,3-benzoxadiazole
3-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)-N-methylpyridin-2-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
1-{1'-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
ethyl 3-(2-phenoxyethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxylate
1-(carbamoylmethyl)-N-methyl-N-(quinolin-8-ylmethyl)piperidine-3-carboxamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl][3-(methylsulfanyl)propyl]amine
N-({7-[(2,5-dimethoxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-4-(4-fluorophenyl)-1-(1H-indol-7-ylmethyl)piperidin-3-ol
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
2-methyl-7-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}butan-1-one
1-ethyl-2-oxo-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}-1,2-dihydropyridine-4-carboxamide
(3S,5S)-1-(3-methylfuran-2-carbonyl)-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
(3S,4S)-4-cyclopropyl-1-[(5-methylpyrazin-2-yl)methyl]pyrrolidine-3-carboxylic acid
methyl 4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}benzoate
4-(2-fluorophenyl)-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-chlorophenyl (7R,9aR)-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-one
(4aS,8aR)-6-[3-(2-fluorophenyl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
ethyl 3-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N4-ethyl-N2-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
2-acetyl-8-(2-methanesulfonylethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
(3S,4S)-1-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-[(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]pyrimidine
2-{5-[6-amino-5-cyano-4-(4,5-dimethylfuran-2-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
1-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(3-methoxypropanoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-cyclopentyl-1-[4-(4-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
3-(3-fluorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-4-carboxamide
1-{5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
methyl (2S,3S)-2-({3-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)-3-methylpentanoate
N-[4-(4-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
2-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-(2,6-dimethoxypyridine-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-2-yl)pyridine
1-{2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
3-(1H-1,3-benzodiazol-2-yl)-N-[2-(2-methoxyethoxy)phenyl]azetidine-1-carboxamide