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8-[(3,5-dimethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]pyridine-3-carbonitrile
(3S,4R)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-cyclopentyl-3-(1-ethyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
2-{2-[6-amino-5-cyano-4-(1-ethyl-1H-pyrazol-4-yl)pyridin-2-yl]phenoxy}acetamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-(prop-2-en-1-yl)-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-1H-indole-2-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-N-(2-methylphenyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(2-methylphenyl)piperidin-1-yl]propan-1-one
3-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-3,9-diazaspiro[5.6]dodecan-10-one
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(5-phenoxyfuran-2-carbonyl)piperidine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
1-(furan-2-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-1-(1,2,3-thiadiazol-5-yl)urea
4-[2-(1H-pyrazol-1-yl)ethyl]-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
1-{1-[1-(2,8-dimethylquinoline-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3,5-dimethyl-4-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
2-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl)benzoic acid
(isoquinolin-5-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-6-(3-methylphenyl)pyridine-3-carboxylic acid
(1S,5R)-3-[2-(2-methoxyphenyl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
N-cyclopropyl-5-[(3-hydroxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(benzyloxy)ethan-1-one
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-({1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methyl)acetamide
4-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
1-{3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}azepan-2-one
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(3-methylpyridin-4-yl)piperazine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine-3-carboxamide
1-({5-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
N,N-diethyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-(2,3-dihydro-1H-inden-2-yl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
8-(3-hydroxybenzoyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({3-[(3-hydroxyazetidin-1-yl)sulfonyl]phenyl}formamido)-N,N-dimethylbutanamide
N-cyclohexyl-3-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)formamido]propanamide
2-hydroxy-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-3-carboxamide
2-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
2-cyclopentyl-2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
3-(1-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(3-methoxyphenyl)-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
1-{2-[4-(4-methylphenoxy)piperidin-1-yl]ethyl}-1H-indazole
4-[(2-oxopyrrolidin-1-yl)methyl]-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide