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1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-ol
9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{4-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
4-{[({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
2-amino-7-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[3-(4-methylpiperazin-1-yl)propyl]-3-(2-methylquinolin-5-yl)urea
3-methyl-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2R,6R)-11-methoxy-4-[(4-methoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(carbamoylmethyl)-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}piperidine-3-carboxamide
2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazole
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[(4-fluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-2-methyl-5-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-2-(4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
2-[8-(1-benzothiophene-5-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
(3S,4S)-3-hydroxy-4-[methyl({[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N4-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-6-methylpyrimidine-2,4-diamine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-[(dimethylamino)methyl]azepan-4-ol
N-[1-(pyridin-3-yl)propan-2-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N3-cyclooctyl-N5-[(2-methoxyphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-1-(2-aminoethyl)-6-[(2E)-3-phenylprop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
N-{1-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
4-[(5-methylfuran-2-yl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
N-cyclooctyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-1-(2-methoxyethyl)-1H-imidazole
3-(2-phenoxyethyl)-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-3-(thiophen-2-yl)propan-1-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[3-(2-methylpropyl)-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl]pyridine
(3S)-2-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylic acid
15-methyl-13-oxo-N-(prop-2-en-1-yl)-9-(pyridin-2-yl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
6-{[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-N-methyl-1,3-thiazol-2-amine
3-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)-6-methoxy-1,4-dihydroquinolin-4-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazinan-2-yl)propanamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]prop-2-ene-1-sulfonamide
(3S,4R)-3-(dimethylamino)-N-[3-(methylsulfanyl)phenyl]-4-propylpyrrolidine-1-carboxamide
1-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-[(3-methylthiophen-2-yl)methyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-(pyridin-2-ylmethyl)urea
N-(2-methyl-1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxolane-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(thian-4-yl)piperidin-4-yl]propanamide
3,6-dimethyl-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
(3aR,6aS)-5-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-chlorophenyl)methyl]-1-ethyl-N-(2-methoxyethyl)piperidine-2-carboxamide
1-[2-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
3-amino-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
3-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]-2,3-dihydro-1λ6-thiophene-1,1-dione