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7-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-(1H-pyrazol-1-yl)-N-(quinolin-5-ylmethyl)benzamide
[5-(4-cyclopentylpyrimidin-2-yl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-3-carboxamide
3-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)phenyl]prop-2-yn-1-ol
2-hydroxy-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)-6-(trifluoromethyl)pyridine-3-carboxamide
2-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[3-(morpholine-4-carbonyl)benzenesulfonyl]-1,4-oxazepane
2,3-dioxo-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrazole
2-[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
8-fluoro-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}quinoline
5-[5-(morpholine-4-carbonyl)furan-2-yl]-1,2,3,4-tetrahydroisoquinoline
3-{2-amino-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl}-1-methyl-1,2-dihydroquinolin-2-one
1-{2-[(2,4-dimethoxyphenyl)formamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2E)-1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(pyridin-2-yl)prop-2-en-1-one
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)pyridine-2-carboxamide
N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(4-acetylphenyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-(1H-pyrazol-1-yl)benzamide
5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-[3-(2-ethoxyphenyl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-methyl-1-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-3-[3-(oxolan-2-yl)propyl]urea
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
3-cyclopropyl-1-[4-(difluoromethoxy)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
1-butyl-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
N-(2-methoxyethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(4-methanesulfonylphenyl)-5-[2-(piperidin-2-yl)ethyl]phenol
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-methylpiperidin-2-one
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(3-methylphenyl)piperidine-1-carboxamide
N-({1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
2-[1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]benzoic acid
(1S,3R)-3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]cyclohexan-1-amine
N-{4-methoxy-3-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}acetamide
{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]azepan-2-yl}methanol
N-[(3R,4S)-4-cyclopropyl-1-[3-(furan-2-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridin-3-ol
1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(propylamino)ethyl]pyrrolidin-2-one
(3aR,6aR)-2-methanesulfonyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 1-(2-methoxyethyl)-5-[2-(pyridin-3-yl)quinoline-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-6-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidine-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
6-ethyl-1,5-dimethyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
5-chloro-2-methoxy-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzene-1-sulfonamide
6-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}pyridine-2-carboxylic acid
1-ethyl-4-{[methyl({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrrolidin-2-one
methyl 5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-1,3-oxazolidin-2-one
(2R,3R,6R)-5-(2,4-dimethylpyrimidine-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-7-fluoro-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
2-{[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]methyl}-8-methoxyquinoline