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2-{[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-5-methylphenol
3-methyl-1-(1-methyl-1H-imidazole-2-carbonyl)-3-phenylpiperidine
1-[(4aR,8aS)-1-(5-fluoro-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
5-butyl-4-(2-methoxyacetyl)-1-(3-phenylphenyl)piperazin-2-one
2-{[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]sulfonyl}benzonitrile
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)-N-methylacetamide
1-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-(1-ethylpiperidin-4-yl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
8-[4-(pyrrolidin-3-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-({5-hexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]propanamide
1-[1'-(4-cyclopentylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(4-aminopiperidin-1-yl)sulfonyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
[2,2-dimethyl-3-(morpholin-4-yl)propyl](1H-imidazol-2-ylmethyl)methylamine
3-chloro-N-cyclopentyl-4-{[1-(prop-2-en-1-yl)piperidin-4-yl]oxy}benzamide
N-{4-[({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}carbamoyl)methoxy]phenyl}propanamide
4-(1H-pyrazol-3-yl)-N-(thiophen-3-ylmethyl)benzamide
5-methyl-3-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-indole
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
2-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-(3-methyl-1-oxo-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-2-yl)acetamide
2-{[4-(pyrimidin-5-yl)phenyl]sulfanyl}acetamide
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-fluorophenyl)piperazin-2-one
4-[5-(3-phenoxypropanamido)-1H-pyrazol-1-yl]-N-(propan-2-yl)piperidine-1-carboxamide
N-benzyl-4-methoxy-4-phenylpiperidine-1-sulfonamide
1-(4-tert-butylphenyl)-3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}urea
4-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
4-[7-(2,5-dimethylfuran-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
2-ethyl-N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)butanamide
1-[(4-methylphenyl)methyl]-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperazin-2-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-carbamoylcyclopropanecarbonyl)pyrrolidine-3-carboxylic acid
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N,N-dimethyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
7-methoxy-N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(2-hydroxybutyl)sulfamoyl]-N-(2-methanesulfonylethyl)benzamide
2-{2-[2-(3-methoxyphenoxy)ethyl]phenoxy}-N-methylacetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2,6-difluorobenzoyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(3S,9aR)-3-benzyl-8-(3,5-dichlorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-(piperidin-3-yl)benzamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-ol
2-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-6-ethoxyphenol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide