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1-[3-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
2-cyclohexyl-1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]ethan-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
3-(3-methoxyphenyl)-5-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)ethan-1-ol
(4aR,7aS)-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-(1H-imidazol-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl (2S)-1-{3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanoyl}pyrrolidine-2-carboxylate
(3S,4R)-1-cyclopentanecarbonyl-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(pyridin-2-ylsulfanyl)propanamide
5-methyl-N-(4-phenylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[4-(4-methoxyphenyl)butanoyl]-1-phenylpiperazin-2-one
7-fluoro-2-methyl-4-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]quinoline
N-methyl-2-(methylamino)-N-(naphthalen-1-ylmethyl)pyridine-3-carboxamide
2-[3-oxo-9-(3-propyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
1-[2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(3aR,7aS)-2-(5-propyl-1,2-oxazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1'-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
4-[(8-chloroquinolin-2-yl)methyl]-N-cyclopropylpiperazine-2-carboxamide
2-[2-(4-phenylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[4-(propylcarbamoyl)phenyl]pyrrolidine-1-carboxamide
4-({4-phenyl-5-[(pyrrolidin-3-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)piperidine
2-ethoxy-3-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
9-(1,5-dimethyl-1H-indazole-3-carbonyl)-3-oxa-9-azaspiro[5.5]undecane
1-(2-{[5-(3-methoxyphenyl)furan-2-yl]formamido}ethyl)piperidine-3-carboxamide
[2-(propan-2-yloxy)-5-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenyl]methanol
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
4-(1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-methylpropan-2-yl)morpholine
4-[1-(1,4-dioxan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-ethoxyphenol
1-[2-(2-chloro-6-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
N-(2-hydroxyethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
5-methyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4,4,4-trifluoro-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]butan-1-one
6-(azepan-1-yl)-N-(2-methoxyethyl)-N-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(2-methylpropyl)-1,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}morpholine
1-methyl-5-(pyrrolidin-1-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
3-(1H-pyrazol-1-yl)-N-[3-(pyridin-2-yl)propyl]benzamide
N-[(3S)-1-[2-(morpholine-4-carbonyl)pyridin-4-yl]pyrrolidin-3-yl]acetamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-(2-fluorophenyl)propyl]-2-(pyrrolidin-3-yl)acetamide
3-cyclopropyl-1-(2,3-dimethylphenyl)-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole