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N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
3-(2,4-difluorophenyl)-1-[2-(dimethylamino)ethyl]-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[(3,4-dimethoxyphenyl)methyl]-5-(2,6-dimethylphenoxymethyl)-1,2,4-oxadiazole
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-(3-propoxypiperidin-1-yl)pyridine
3-{[(2-chloro-6-fluorophenyl)methyl](cyclopropyl)carbamoyl}benzoic acid
(3aS,6aS)-2-(furan-3-carbonyl)-5-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-cyclopropanecarbonyl-1'-(3-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-N-methylpyridine-3-carboxamide
(2S,4R)-1-benzyl-N,N-diethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(3R,5S)-N-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
5-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-N,N-dimethylpyrimidin-2-amine
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)benzamide
(1S,5R)-6-(oxane-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
N5-cyclopentyl-1-(2-methylpropyl)-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2S,4S)-4-amino-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]pyrrolidine-2-carboxylic acid
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]benzene-1,3-diol
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-2-(4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
methyl (2S,4R)-1-methyl-4-[1-(pyrimidin-2-yl)piperidine-4-amido]pyrrolidine-2-carboxylate
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(cyclopropylmethyl)pyrrolidine-2-carboxamide
ethyl 1-[2-(4-hydroxy-2,6-dimethylpyrimidin-5-yl)acetyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}pyrimidin-4-amine
5-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
5-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-oxo-1-(pent-2-yn-1-yl)-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-{3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-5-{[(9H-fluoren-2-ylmethyl)amino]methyl}phenyl}acetamide
2-(benzyloxy)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
2-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl 6-(1-methyl-1H-pyrazole-5-carbonyl)-2-{[(4-methylphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-fluorophenyl)-N-methyl-N-(oxan-4-yl)imidazo[1,2-a]pyridine-6-carboxamide
ethyl 2-[({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]acetate
(4aR,7aS)-1-cyclopropanecarbonyl-4-(4-methoxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-methyl-3-phenylpiperidin-1-yl)-6-(pyrrolidine-1-carbonyl)pyrazine
4-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}morpholine
(2S,4S)-4-amino-1-[3-(prop-2-en-1-yloxy)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
5-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}isoquinoline
1-ethyl-8-[(2E)-2-methylbut-2-en-1-yl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[4-(3-ethoxyphenyl)thiophen-2-yl]methyl}piperazine
3-({3-[3-(pyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)benzonitrile
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1-phenylpropyl)propanamide
7-(3-chlorophenyl)-4-(piperidin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-4-(pyridin-2-yl)piperazine
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one