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2-(3-{3-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
(3R,4S)-4-cyclopropyl-1-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-amine
1-ethyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-fluorophenyl)pyridine-3-carboxylic acid
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1-methylpiperidin-4-yl)piperazine
4-[3-(3-chlorophenyl)-3-(3-hydroxyphenyl)propanoyl]-3,3-dimethylpiperazin-2-one
1-[benzyl(methyl)amino]-3-[4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-(3-hydroxy-3-methylbutyl)-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]benzamide
3-chloro-5-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-{[(1,3-dihydroxy-2-methylpropan-2-yl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(3-fluoro-4-methylphenyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
3-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,2-dihydroquinoxalin-2-one
6-methyl-N4-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]pyrimidine-2,4-diamine
N-(2,3-dihydroxypropyl)-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)piperidin-2-one
3-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
6-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-ol
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
N-(1,3-dihydro-2-benzofuran-5-yl)-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(1S,5R)-3-(6-methylpyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-4-cyclopentylpyrimidin-2-amine
4-hydroxy-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-(methoxymethyl)benzamide
1-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)azepan-4-amine
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-{1-[(2-phenylphenyl)methyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(oxane-4-carbonyl)piperidine
3-methyl-3-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
ethyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1-(4-tert-butylphenyl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-[(1-cyclobutylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(oxolan-2-ylmethyl)amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{[6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyrimidin-4-yl]amino}ethan-1-ol
2-(4-fluorophenyl)-4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}morpholine
1-[cyclopropyl(4-methoxyphenyl)methyl]-3-(1-methyl-1H-1,3-benzodiazol-5-yl)urea
6-ethyl-N4-[1-(furan-2-carbonyl)piperidin-4-yl]-N2,N2-dimethylpyrimidine-2,4-diamine
4-[3-(azocan-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
1-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(1,2-oxazolidin-2-ylmethyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-1,8-naphthyridine-2-carboxamide
N-(dicyclopropylmethyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
5-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1,3,4-thiadiazol-2-amine
1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(1-methoxypropan-2-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide