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N-ethyl-7-fluoro-2-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]quinoline-4-carboxamide
1-[(1-methylpiperidin-4-yl)methyl]-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazine
2-(2-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}quinolin-8-ol
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2,4-dimethoxybenzamide
2-tert-butyl-5-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidin-4-ol
2-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
13-[3-(2-methylphenyl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
4-[2-(methylsulfanyl)phenyl]-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-1-(3,5-dichloro-4-methylbenzoyl)-octahydropyrrolo[2,3-c]pyrrole
2-{[5-(4-ethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
8-{[3-chloro-4-(prop-2-yn-1-yloxy)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-{2-[(4-methoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethylpiperidin-3-ol
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
9-(1-ethyl-1H-1,2,4-triazol-5-yl)-2H,3H,6H,7H,8H,9H-[1,4]dioxino[2,3-g]quinolin-7-one
1-[3-(5-methyl-1H-pyrazol-1-yl)propyl]-4-(pyridin-2-yl)piperazine
N-(2-methoxyethyl)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
N-cyclopentyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
2-(1-methylpyrrolidin-3-yl)-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-acetyl-8-(4-methoxy-3-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclopropyl-1-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-(hydroxymethyl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]azepan-4-ol
2-(2-chlorophenyl)-3-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-(3-chloro-4-fluorobenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(3R,4R)-1-(benzenesulfonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-[2-(2-fluorophenyl)ethyl]-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
3-chloro-4-hydroxy-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
N,1-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-{[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl](methyl)amino}pyrimidine-5-carboxylic acid
N-cyclohexyl-2-[(3,4-dimethoxyphenyl)methyl]-N-(prop-2-yn-1-yl)-1,3-benzoxazole-6-carboxamide
2,4-dimethyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
3-(5-methylfuran-2-yl)-5-(pyrrolidin-3-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
6-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine
2-[3-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-indol-1-yl]acetamide
3-(2-fluorophenyl)-N-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidine
3-(3,5-dimethylphenyl)-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
2-[2-(dimethylamino)ethyl]-8-[2-(pyrazin-2-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2,7,8-trimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]quinoline-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]acetamide
2-(1-ethylpiperidin-4-yl)-N-[1-(4-fluorophenyl)-2-hydroxyethyl]acetamide
2-{2-methylimidazo[2,1-b][1,3]thiazol-6-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(isoquinolin-5-ylmethyl)-N-methyl-1-benzoxepine-4-carboxamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(1-methyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-1-yl]acetamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide