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6-(2-ethoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-benzyl-4-[1-(oxolane-3-carbonyl)piperidin-4-yl]piperazine
4-[4-(4-chlorophenyl)-5-ethyl-1H-imidazol-2-yl]-1-cyclopentylpyrrolidin-2-one
14-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-ethyl-1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidine-3-carboxamide
ethyl 5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-1-(1,5-dimethyl-1H-pyrazole-4-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-(1-benzylcyclopropyl)-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-hydroxy-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]pyridine-2-carboxamide
2-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
methyl (2S,4S)-4-(2-cyclopentylacetamido)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
6-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
1,5-dimethyl-4-(5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1H-pyrazole
8-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-(3-methylthiophen-2-yl)-1H-imidazole
1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
4-(1-benzothiophen-3-yl)-6-(methoxymethyl)pyrimidine
5-(2-chloro-4-fluorophenoxymethyl)-N-(3-hydroxy-2,2-dimethylpropyl)-1,2-oxazole-3-carboxamide
4-(2-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)phenol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
2-methyl-5-{1-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}pyridine
4-[4-(piperidin-1-yl)benzoyl]piperazine-1-sulfonamide
N4-[(2,6-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
4-[3-(carbamoylmethyl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
1-(3-methoxyphenyl)-4-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperazin-2-one
1-(5-fluoro-1H-indole-2-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
1-{4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]phenyl}-1H-pyrazole
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
3-(3,4-difluorophenyl)-5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
ethyl 4-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
7,11-dimethyl-3-(pyridin-4-ylmethyl)-3,7,11-triazaspiro[5.6]dodecane
4-(3-methylphenoxy)-N-(4-sulfamoylphenyl)piperidine-1-carboxamide
1-[1'-(morpholine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
methyl 3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
1-{[4-(methylsulfanyl)phenyl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-ethylpyridine-3-carboxamide
(2S,4S)-4-amino-1-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-N-methylpyrrolidine-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
3-cyclobutyl-5-(3-fluoro-4-methoxyphenyl)-1H-1,2,4-triazole
1-butyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
ethyl 2-amino-3-cyano-4-(3-ethyl-1H-pyrazol-5-yl)-5,6,7,8-tetrahydroquinoline-6-carboxylate
1-benzyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-4-amine
1-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-3-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N3-[3-(benzylsulfanyl)propyl]piperidine-1,3-dicarboxamide
8-acetyl-2-[(3-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid