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3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
(2S,4S)-4-amino-1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
(3R,5R)-N-(2-methylpropyl)-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
(3R,4R)-1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-4-ethylpiperidine-3,4-diol
1-(4-cyanopyridin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
4-(2,2-dimethylpropyl)-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-({2-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]phenyl}methyl)propanamide
N'-[2-(4-cyclooctylmorpholin-2-yl)ethyl]ethanediamide
3-[(4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
4-({2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2,3-dimethyl-7-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-chloro-4-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
3-{[ethyl(oxan-4-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[2-(5-methylthiophen-2-yl)ethyl]urea
5-(1-methanesulfonylpyrrolidine-2-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1R,3S)-3-methoxy-7-(5-methoxyfuran-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-(2-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-(1,2,3,4-tetrahydroisoquinolin-2-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
{2-[(5-ethylpyrimidin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
4-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-phenylpiperidin-1-yl)acetamide
1-(4-methoxyphenyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
4-(4-cyclohexylpiperazine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2-methylpropyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[5-(5-cyclopropyl-1,3-oxazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
6,7-difluoro-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
(2R)-2-amino-4-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pentanamide
4-{4-[(5-chloro-2-hydroxyphenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
5-[(furan-2-ylmethyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3,5-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-({1-[2-(1H-imidazol-4-yl)acetyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
2-(dimethylamino)-8-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-cyclobutyl-N-[(3R,4S)-4-cyclopropyl-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl]acetamide
1-benzyl-5-(butylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(1-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-oxopropan-2-yl)sulfanyl]-6-methyl-3,4-dihydropyrimidin-4-one
3-(naphthalen-1-yl)-5-(oxane-4-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
(2-{2-[1-(benzenesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N,N-dimethyl-5-[3-(1-methylpiperidin-3-yl)propanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-(2,4-dimethoxyphenyl)-1-(2-hydroxyethyl)-1-[(2-methylphenyl)methyl]urea
(2S)-3-(1H-indol-3-yl)-2-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)propanoic acid