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(4aS,7aR)-1-[2-(4-fluoro-3-methylphenyl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-tert-butyl-6-(3-chloro-5-fluorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-[4-(5-{[(2-methylphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetamide
(1R,5R)-6-(3-hydroxypyridine-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-(2-hydroxyethyl)-N-(naphthalen-1-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(furan-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
N-(1H-imidazol-2-ylmethyl)-N,4-dimethyl-2-phenylpyrimidine-5-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-(furan-2-ylmethyl)-N'-(2-methylphenyl)-N-(prop-2-en-1-yl)propanediamide
1-(azocan-1-yl)-3-{5-[(cyclohexylamino)methyl]-2-methoxyphenoxy}propan-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-({3-[(5-methylpyridin-2-yl)amino]propyl}amino)propan-1-ol
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(dimethylamino)ethan-1-one
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(2-methylpropanoyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
3-(2-chlorophenoxy)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}azetidine
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-[(2-methyl-1,3-benzothiazol-5-yl)methyl]-1λ6-thiane-1,1-dione
N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]azepane-1-carboxamide
4-(2-methoxyethoxy)-1-{[2-(methylsulfanyl)phenyl]methyl}piperidine
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
2-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-cyclohexyl-1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]propan-1-one
4-(3-hydroxy-3-methylbutyl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-ethyl-N-methyl-6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-3-carboxamide
N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-1,2,3-triazole-5-carboxamide
2-(2-aminopyrimidin-5-yl)-3,6-dimethyl-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
6-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}methyl)pyrimidin-4-ol
4-{5-[3-(ethylsulfanyl)phenyl]furan-2-carbonyl}morpholine
4-(1-ethyl-1H-imidazol-2-yl)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
1-(2H-1,3-benzodioxol-5-yl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
2-{[5-fluoro-2-(4-methoxy-2,6-dimethylphenyl)pyrimidin-4-yl]amino}ethan-1-ol
6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
9-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}propanamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
2-[(dimethylamino)methyl]-N-ethyl-N-{[4-(propan-2-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
1-(1-{1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3aR,7aS)-2-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(1s,4s)-4-hydroxy-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]cyclohexane-1-carboxamide
2-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-methyl-1,3,4-oxadiazole
8-(3-hydroxypyridine-2-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
2-amino-6-(4-chloro-3-methylphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
1-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one