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N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(2-fluorophenoxymethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1,3-oxazole-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-[(2S)-1-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
3-(5-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
(4aS,7aR)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-1-(4-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)pyrrolidine-2-carboxylic acid
5-tert-butyl-4-[(2-oxo-1,2-dihydroquinolin-1-yl)methyl]furan-2-carboxamide
6-[2-(morpholin-4-ylmethyl)phenyl]pyridine-3-carboxylic acid
2-methoxy-4-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
2-(3-hydroxypropyl)-8-[(1-methyl-1H-indol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methoxy-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
ethyl 1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-(5-ethyl-1H-pyrrole-2-carbonyl)-3-methyl-3-phenylpiperidine
1-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-2-yn-1-one
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(4-ethoxy-2-fluorophenyl)urea
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4-methylpyrimidin-2-amine
2-(1-methyl-1H-pyrazol-4-yl)-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
6,7-dimethyl-2-(1,2,3,6-tetrahydropyridin-1-ylmethyl)-1H-1,3-benzodiazole
1-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}butan-2-ol
4-[1-(1-methylpiperidin-4-yl)-5-(2-phenoxyethyl)-1H-1,2,4-triazol-3-yl]pyridine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(4-methylphenoxymethyl)piperidine
8-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{1-[2-(piperidin-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
7-methyl-2-(quinoxalin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-2-{4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperazin-1-yl}acetamide
3-(1H-1,3-benzodiazol-2-yl)-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole
N-(4-methoxy-2-methylphenyl)-2-(3-methoxypropyl)piperidine-1-carboxamide
N3-[1-(4-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(2-{4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3-oxazolidin-2-one
2-(propylsulfanyl)-5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
1-{[2-(pyrimidin-2-yl)phenyl]methyl}piperidin-4-one
3-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}-N-(2-fluoro-5-methylphenyl)propanamide
9-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-{[(2-{5-oxo-1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
[1-({1-[(5-ethylthiophen-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
(2R,3R,6R)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,6S)-2,6-dimethyl-4-{1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}morpholine
4-{[ethyl(propan-2-yl)amino]methyl}-N-(6-methylpyridazin-3-yl)benzamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
1-methyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]imidazolidin-2-one
N-(3-chloro-4-methoxyphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-methyl-4-(pyrimidin-2-ylmethyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
5-cyclohexaneamido-N-(2,3-dihydro-1H-inden-1-yl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
6-{[(1R)-1-carbamoyl-2-methylpropyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-[(1-methyl-1H-imidazol-2-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one