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5-{1-[(4-chlorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-{4-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]phenyl}-5-methyl-4H-1,2,4-triazole
4-ethyl-3-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[1-(4-methylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
(3S,4S)-4-cyclopropyl-1-{[2-(2-hydroxyethoxy)phenyl]methyl}pyrrolidine-3-carboxylic acid
(1S,5R)-6-(1H-indole-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-({[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}(methyl)amino)-N,N-dimethylpropanamide
8-(6-tert-butyl-2-oxo-2,3-dihydropyrimidine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-(1,2-oxazolidin-2-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
4-{[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]methyl}morpholine
N,N-dimethyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-1,2,3-triazole
2-(dimethylamino)-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
1-[(furan-2-ylmethyl)carbamoyl]-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
4-{2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
6-ethyl-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2-methylquinoline
2-{[(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
5-{[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
1-[2-(1H-imidazol-1-yl)ethyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
2-({[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-8-fluoroquinolin-4-ol
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-(2-hydroxyethyl)piperazin-2-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N-[(4-methoxyphenyl)methyl]-5-(3-methylbutanoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanoic acid
N'-(3-chloro-4-fluorophenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]butanediamide
N-[1-(methoxymethyl)cyclopentyl]-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
5-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
5-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridine-3-carboxamide
1-[3-(furan-2-yl)propyl]-2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazole
(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
ethyl({[2-(2-methylphenyl)pyrimidin-5-yl]methyl}){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
9-[(1-propyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-[1-(thiophen-2-yl)butyl]-2-(thiophen-2-ylformamido)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-[(4-cyclopentylpyrimidin-2-yl)amino]-N-methylbutanamide
N-cyclopropyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}benzamide
4-(5-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-yl)morpholine
2-fluoro-5-sulfamoyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
5-fluoro-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]quinazoline
1-[(4aR,8aS)-1-(2-methoxybenzoyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-[2-(benzyloxy)ethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
4-(4-chlorophenoxy)-1-(3-hydroxybenzoyl)piperidine-4-carboxylic acid
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-phenyl-1,2,3,6-tetrahydropyridine
2-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one