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N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3-chlorophenyl)-4-[(2-methoxypyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-ethyl-2-(piperidin-1-yl)-N-(pyridin-2-ylmethyl)pyrimidin-4-amine
butyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-cyclopentyl-4-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)-5-methylpyrimidin-4-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(propan-2-yl)piperidine-3-carboxamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4-difluorophenyl)methyl]piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-fluoro-N-methylquinazolin-4-amine
(4aS,8aR)-1-(2-phenylethyl)-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-amino-7-(1-propyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{2-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(3-methylbutyl)-3-(propan-2-yl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
1-(3-methylbutyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2-fluoro-5-methoxyphenyl)methyl]amino}pyrrolidin-2-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
4-{[(6-methylpyridin-2-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(2,3-dimethylphenoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1R,5R)-6-[(2,4-dimethoxyphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2R,3R)-2-methoxy-1'-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-[3-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(3-methylphenyl)methyl]piperazine
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-(2,2-dimethylpropyl)piperidin-4-ol
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
N-cyclopentyl-2-(4-cyclopropyl-4-methyl-2-oxopyrrolidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
2,7-dimethyl-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-ethyl-2-[4-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperazin-1-yl]acetamide
methyl 2-(diethylsulfamoyl)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[2-(dimethylamino)-4-[(2-phenoxyethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1,4-dimethyl-9-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-1,4,9-triazaspiro[5.5]undecane
1-[(2,4-difluorophenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-cyclopentyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[1-(2-methylphenyl)piperidin-4-yl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-amino-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
3-(hydroxymethyl)-N-(2-methoxy-5-phenylphenyl)morpholine-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-chloropyridine-4-carbonyl)piperidin-3-ol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1-{4-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-1-yl}ethan-1-one
methyl[(5-methylfuran-2-yl)methyl]{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
N-(4-fluoro-3-methylphenyl)-4-(pyrrolidin-1-yl)piperidine-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-2-one