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2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-(adamantan-1-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
4-(1H-imidazol-1-yl)-1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidine-4-carboxylic acid
2-{[2-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
3-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-N-[(4-fluorophenyl)methyl]propanamide
N-methyl-3-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-N-(1-methylpiperidin-4-yl)propanamide
4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)benzoic acid
4-{1-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
9-(2-methoxyethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-(2-butoxy-4-fluorophenyl)-6-(4-methylpiperazin-1-yl)pyridazine
3-(3-methyl-1-propyl-1H-pyrazol-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
[(3R,4S)-1-{[4-(2-methylpropyl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-(thiophen-3-yl)acetamide
5-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(4-methyl-1,4-diazepan-1-yl)-2-[2-(propan-2-ylsulfanyl)ethyl]-2,3-dihydropyridazin-3-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)benzamide
ethyl 4-[4-(4-{[(3-fluoro-4-methylphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-butyl-4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methylpiperazin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-[(4-phenyloxan-4-yl)methyl]-6-(1,3-thiazol-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butane-2-sulfonamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(2-methylpropyl)benzamide
4-hydroxy-2-methyl-N-[3-(pyridin-2-yl)propyl]benzamide
3-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperazin-1-yl)-2,5-dimethylpyrazine
8-[4-methoxy-3-(morpholin-4-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxan-2-ylmethyl)acetamide
2-(3-hydroxypropyl)-9-(2-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(pyrrolidin-1-ylmethyl)piperidine
(3R,5S)-N-methyl-5-(morpholine-4-carbonyl)-N-[2-(phenylsulfanyl)ethyl]piperidine-3-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
1-methyl-5-(4-methylpiperidin-1-yl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]cyclopropanecarboxamide
2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
2-methyl-8-[2-(pyridin-3-yloxy)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,N,4-trimethyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
2-{[(4-methyl-1H-imidazol-5-yl)methyl][(2-methylphenyl)methyl]amino}ethan-1-ol
2-cyclohexyl-5-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}pyrimidine
4-ethyl-1-methyl-3-({1-[2-(1H-pyrazol-1-yl)butanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-chloro-N-[(3R)-piperidin-3-yl]-5-(1H-pyrazol-1-yl)benzamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{2-[(4-methylphenyl)methyl]benzoyl}piperidin-4-ol
1-(propan-2-yl)-4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperazine
8-(3-methoxypyrazin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(adamantan-1-yl)-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
5-methyl-1-{2-oxo-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,7aS)-N,N-dimethyl-4-{[3-(methylsulfanyl)phenyl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(1-methylpiperidin-2-yl)-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]propan-1-one