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1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[2-(4-ethoxy-6-methylpyrimidin-2-yl)phenoxy]thiane-4-carboxylic acid
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-sulfonyl]-N-(pyridin-3-yl)benzamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(2-phenylethynyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-[2-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)ethyl]methanesulfonamide
1-methyl-N-[(5-methylfuran-2-yl)methyl]-5-({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[1-(dimethyl-1,3-thiazole-5-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
2-{1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
(1S,5R)-6-methyl-3-[2-(morpholin-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-2-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl]methanol
4,6-dimethyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carbonitrile
ethyl 5-(1H-indol-3-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(2-methyl-1,3-benzothiazol-6-yl)-1-[(3R)-pyrrolidin-3-yl]urea
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-ethyl-N-methylpyrimidine-5-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)but-2-enamide
2,4-dimethyl-5-[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)carbamoyl]-1H-pyrrole-3-carboxylic acid
1-(1,2,3,4-tetrahydroisoquinolin-5-yl)isoquinoline
2-[4-({[2-(1H-indol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-[3-(dimethylcarbamoyl)-5-[({[4-(propan-2-yl)phenyl]methyl}amino)methyl]phenyl]pyridine-2-carboxamide
1,5-dimethyl-4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl 4-(4-{5-methoxy-2-[(2-methoxyethyl)carbamoyl]phenoxy}piperidin-1-yl)pentanoate
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl](4-methoxy-4-methylpentan-2-yl)amine
2-[3-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-[2-(adamantan-1-yl)acetyl]-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
2-[2-(methylsulfanyl)phenyl]-2-(pyrrolidin-1-yl)acetic acid
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-2-hydroxyacetamide
4,6-dimethyl-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2H-pyran-2-one
4-(propan-2-yl)-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(trifluoromethyl)pyrimidine
N-{[3-(trifluoromethyl)phenyl]methyl}morpholine-2-carboxamide
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-(oxan-4-yl)acetamide
N,5-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-(3,5-dimethoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(hydroxymethyl)azepan-4-ol
2-(4-methoxyphenyl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-(3-methoxyphenyl)-4-(2-methoxypyridine-4-carbonyl)piperazin-2-one
N-butyl-3-{4-[(propan-2-yl)amino]pyrimidin-2-yl}benzamide
(1R,5S,8R)-8-methoxy-3-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octane
2-(cyclopropylmethyl)-N-methyl-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)sulfonyl]-N-methylbenzamide
4-[4-(3-chlorobenzoyl)-2-oxopiperazin-1-yl]benzonitrile
ethyl 4-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidine-1-carboxylate
4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-ol
2-{3-[(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(pyrrolidin-3-yl)benzamide
1-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
2-(cyclopentylmethyl)-N,6-dimethyl-4-oxo-1-(pyridin-3-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine