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1-[(6-methylpyridin-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(1-methyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
3,5-difluoro-2-[4-(1-methylpiperidin-4-yl)piperidine-1-carbonyl]pyridine
2-({4-[3-(1-methylpiperidin-2-yl)propanoyl]piperazin-1-yl}methyl)benzonitrile
1-(cyclopentylcarbamoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
9-{2-[4-(dimethylamino)phenyl]acetyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoline
1-[4-(3-methoxyphenyl)phenyl]-N-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-amine
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)methanesulfonamide
5-methoxy-2-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-4H-pyran-4-one
1'-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(4-fluoro-2-methylphenyl)-3-({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propanamide
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-(1H-imidazol-2-yl)piperidine
2-(cyclohex-1-en-1-yl)-N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(6-methylpyridin-2-yl)piperazine
(3S,4R)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-methyl-N-[3-(morpholin-4-yl)propyl]-5-(3-phenylprop-2-ynoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
1-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
3-[1-(5-propyl-1,2-oxazole-4-carbonyl)azetidin-3-yl]pyridine
N-(4-methoxy-3-propanamidophenyl)-3-phenylpiperidine-1-carboxamide
2-(6-aminopyridin-3-yl)-2-{[2-(dimethylamino)ethyl](methyl)amino}acetic acid
2-{5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[(4-fluorophenyl)methyl]-3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]propanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-(2-hydroxyethyl)-N-methyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-(3-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-3-phenylpropanamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxo-2-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
N,1,6-trimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-5-chloro-3-phenyl-1H-indole-2-carboxamide
(2S,4S)-4-amino-1-(5-chloro-2-methoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-ethyl-N-[(2-fluorophenyl)methyl]-1H-pyrazole-3-carboxamide
ethyl 1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxylate
1-cyclopentyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(2,2,6,6-tetramethylpiperidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-acetyl-8-(1-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(3-methoxyphenyl)methyl]piperidine
3-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
6-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,2-dimethylquinoline-4-carboxamide
1-[2-(ethylsulfanyl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-(5-methyl-1,2-oxazol-3-yl)-2-(4-methylpyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-[2-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide