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N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(oxolan-2-ylmethyl)piperidin-4-amine
2-{1-[(2-methylphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[1-(2,5-dimethylphenyl)ethyl]-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
N-[(3R,4S)-4-cyclopropyl-1-(6-methoxypyrimidin-4-yl)pyrrolidin-3-yl]oxane-4-carboxamide
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
(4S)-3,3,4-trimethyl-1-(pyrimidin-2-ylmethyl)piperidin-4-ol
2-methoxy-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methoxy-6-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
N-[(2R,3R)-1'-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
2-(4-{[2-(methoxymethyl)piperidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
2-{4-[(4-chlorophenyl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
methyl 1-[(3S,5S)-1-cyclopentyl-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyridazin-3-amine
N'1-(2-methylpropyl)-N'1-(thiophen-3-ylmethyl)cyclopropane-1,1-dicarboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}propanamide
N-[4-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}sulfonyl)phenyl]acetamide
2-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
3-(2,3-dimethoxy-5-methylphenyl)-N-methylbenzamide
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-(propan-2-yl)-2-[5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1H-1,3-benzodiazole
N-[(3R,4R)-3-hydroxy-1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
1-(benzylsulfamoyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
(3aR,6aR)-2-cyclopentyl-5-[(4-methyl-1,3-thiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
1'-(1-benzoxepine-4-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-ethylbutan-1-one
3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
2-({[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-6-fluoroquinolin-4-ol
2-(2-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(4aS,8aR)-2-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-decahydroisoquinoline
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylthiophene-2-carboxamide
5-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(4-oxo-1,4-dihydropyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl N-(1-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1-oxopropan-2-yl)carbamate
ethyl 1-{2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetyl}piperidine-3-carboxylate
[(3R,4R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-propylpiperidin-3-yl]methanol
2-(morpholin-3-yl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)acetamide
1-({1-[(1-methanesulfonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)azepane
(1S,3R)-N-(2,3-dihydro-1H-inden-5-yl)-3-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]cyclopentane-1-carboxamide
4-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}-2-methylbutan-2-ol
1-(3-methoxyphenoxy)-3-(4H-1,2,4-triazol-4-yl)propan-2-ol
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylphenyl)methyl]acetamide
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-({5-[1-(2-amino-2-methylpropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol