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N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methylquinoline-4-carboxamide
2-(2-ethylphenyl)-2-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid
3-[3-({[(1S)-2-hydroxy-1-phenylethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
4-ethyl-2-methyl-6-{4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-(oxolan-2-ylmethyl)acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(pyridin-4-yl)piperidin-3-yl]propanamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-9H-fluorene-9-carboxamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-phenylpyrimidin-2-amine
4-methoxy-N-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1,9-dimethyl-4-(3-phenoxypropanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(7-chloro-1-methyl-1H-indole-2-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-(3-butoxyphenyl)-4-cyclopentyl-3-oxopiperazine-1-carboxamide
6-methyl-2-(piperidin-1-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
1-[2-(3-fluorophenyl)ethyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
N-benzyl-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
4-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}-3-methoxyphenol
N-(2-oxooxolan-3-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]phenyl}-2-methylpropanenitrile
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,3-benzoxazol-2-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-methoxy-4-oxo-4H-pyran-2-carboxamide
N-[1-(3-methylpyridin-2-yl)ethyl]-3-(1,2-oxazolidin-2-yl)propanamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4,4,4-trifluorobutan-1-one
(3S,4S)-4-(4-fluorophenyl)-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]piperidin-3-ol
(2S,4R)-4-amino-N,N-diethyl-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
1-[3-(3-methoxyphenyl)propanoyl]-3-methylpiperidine-3-carbonitrile
2-(2-methoxy-4-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)acetamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperidine
methyl (2S,4R)-1-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-4-hydroxypyrrolidine-2-carboxylate
6-[(5,6-dimethylpyrimidin-4-yl)amino]-2-methylheptan-2-ol
(1S,5R)-3-(4-methylpyrimidin-2-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methylthiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
9-(3,4-dimethylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohex-3-ene-1-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-ethyl-N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
5-methyl-1'-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
1-[(3S,4R)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(3aS,6aS)-2-[(4-chloro-2-fluorophenyl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-indazole-3-carboxamide
2-fluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenylacetamide
benzyl 3-{[(5-methylpyrimidin-2-yl)amino]methyl}piperidine-1-carboxylate
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]pyrrolidine-1-sulfonamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(1H-imidazol-1-yl)propyl]acetamide
1-cyclohexyl-N3-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4R)-3-[ethyl({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})amino]-4-hydroxy-1λ6-thiolane-1,1-dione
N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(oxan-2-ylmethoxy)acetamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]thiophene-3-carboxamide
4-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine