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1-[1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-methoxybenzamide
{[5-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 2-{[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]sulfonyl}benzoate
1-[4-(2-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
N-[(3S,4R)-4-methoxyoxolan-3-yl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-cyclopropyl-N-(2-hydroxyethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylpyrazolo[1,5-a]pyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-(1H-pyrrol-1-yl)benzamide
2-(2-phenylethyl)-9-(propane-2-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
N,1-dimethyl-N-(2-methylpropyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(trifluoromethyl)benzamide
N-cyclopentyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-chlorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
2-cyclopropyl-4-hydroxy-N-[2-(5-methylfuran-2-yl)ethyl]pyrimidine-5-carboxamide
2-{3-[1-(oxan-4-ylmethyl)-1H-imidazol-2-yl]phenoxymethyl}pyridine
N6-cyclopentyl-N5-methyl-N5-(oxan-4-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2,3-dimethyl-6-[4-(pyridin-3-yl)pyrimidin-2-yl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
14-(2-hydroxy-6-methoxyquinolin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-[(2-fluorophenyl)methyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
7-[4-(1H-pyrazol-3-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-N-(dimethyl-1,2-oxazol-4-yl)piperidine-1-carboxamide
2-cyclobutyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-1,3,4-oxadiazole
N-[(3,5-difluoro-4-methoxyphenyl)methyl]pyrimidin-4-amine
3-benzyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
2-[5-(azepan-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-[3-(2-methylpropyl)-5-(pyridin-2-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[(2R,4R,6S)-2-cyclohexyl-6-[2-(pyridin-2-yl)pyrimidin-5-yl]oxan-4-yl]acetamide
2-(1H-1,3-benzodiazol-2-ylmethyl)-9-oxa-2-azaspiro[5.5]undecane
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(pyrazin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
5-methoxy-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-4-oxo-4H-pyran-2-carboxamide
4-[2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethyl]morpholine
6-methyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[2-(trifluoromethoxy)phenyl]methyl}amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
2-[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carbonyl]-6-methyl-4H-pyran-4-one
(3aR,5R,6S,7aS)-2-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-octahydro-1H-isoindole-5,6-diol
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
2,2-dimethylpropyl 2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
5-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3,4-dihydropyrimidin-4-one
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,6-difluorophenyl)methyl]piperidine