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(3R,9aR)-8-[(2,4-dimethylphenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-(cyclopropylmethyl)-1-methyl-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-N-(3-ethoxypropyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3aS,6aS)-5-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-N,N-diethyl-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
2,3-dimethyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]quinoxaline-6-carboxamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylacetamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-4-carboxamide
1-[(2-aminopyrimidin-5-yl)methyl]-3-(2,3-dihydro-1H-inden-5-yl)-1-methylurea
3-cyclopropyl-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1H-pyrazole-5-carboxamide
4-methyl-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}quinoline
1-cyclohexyl-N3-[(2,5-difluorophenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(1-{[1-(4-methylbenzenesulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(2S,4R)-4-amino-N-(propan-2-yl)-1-(quinolin-2-ylmethyl)pyrrolidine-2-carboxamide
3-({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}(ethyl)amino)-1λ6-thiolane-1,1-dione
3-(quinoxalin-2-yl)-4H-chromen-4-one
3-({[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]oxy}methyl)pyridine
(3R)-1-(2-methoxybenzenesulfonyl)-3,4,4-trimethylpyrrolidin-3-ol
(4aS,7aR)-1-(6-ethyl-2-methylquinoline-4-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-indazole
N-[(2R)-2-hydroxypropyl]-4-{[2-(3-methyl-1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
N-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-1-ethyl-N-methylpiperidin-4-amine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
4-(1-ethyl-1H-imidazol-2-yl)-1-(1-ethylpiperidine-2-carbonyl)piperidine
2-(5-fluoro-2-methylphenyl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)acetamide
4-[(5-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
2-(2-chloropyridine-4-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
(1R,5S)-3-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,8-diazabicyclo[3.2.1]octane
2-(2-chlorophenoxy)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N6-cyclopropyl-N4-(furan-3-ylmethyl)-N4-methylpyrimidine-2,4,6-triamine
4-{[(2-amino-5-ethylpyrimidin-4-yl)amino]methyl}-N,N-dimethylbenzene-1-sulfonamide
2,6-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyridine-4-carboxamide
1-[1-(oxan-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
1-cyclohexyl-N3-methyl-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
propan-2-yl 7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
(2S)-2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]-3-methylbutanamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[4-(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]ethan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-{2-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-[3-(furan-2-yl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
(3aR,6aR)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-{pyrazolo[1,5-a]pyridin-7-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-[(2,4-dimethoxyphenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea