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1-({5-[(3-fluoro-2,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-cyclopropyl-4-(3-hydroxy-3-methylbutyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(2-fluorophenyl)pyrrolidine
1-{2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-N-methylpyrrolidine-3-carboxamide
2-amino-4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-{1-[2-phenyl-2-(piperidin-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
6-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-phenylpyrimidin-4-amine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
5-({[2-(cyclohex-1-en-1-yl)ethyl](cyclopropylmethyl)carbamoyl}amino)-2-methoxybenzamide
N4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2S,4R)-1-benzyl-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4R)-N-methyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamido]-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
1-benzoyl-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)-N-[2-(prop-2-en-1-yloxy)phenyl]pyrrolidine-1-carboxamide
N-cyclopentyl-4-[(2-oxopyrrolidin-3-yl)sulfamoyl]benzamide
2-hydroxy-S-(4-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}phenyl)propane-1-sulfonamido
2-(methylsulfanyl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide
5-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-2-methylphenol
2-methyl-6-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(2-methylphenyl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3S,4S)-4-methyl-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}pyridin-2-amine
1-ethyl-4-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
4-ethyl-3-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1,7-dimethyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-indole-2-carboxamide
4-{1-[2-(2,4-dimethoxy-3-methylphenyl)-1H-imidazol-1-yl]ethyl}phenol
4-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1-phenylpiperazin-2-one
1-(2-fluorophenyl)-4-[(3-{[1-(pyridine-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
7-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[3-(3-methylphenyl)phenyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
9-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-{2-[4-(3-methoxyphenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
7-(1,3-benzothiazol-2-yl)-4-(2,3-dihydro-1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,5S)-5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-amine
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
6-fluoro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1-(diphenylmethyl)-N,N-bis(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-(3-methoxypropyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]pyridine-2-carboxylic acid
5-[(2-methoxyethyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 3-({[1-(3,4-dimethoxyphenyl)ethyl]carbamoyl}amino)-4-methoxybenzoate
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[3-(4-fluorophenoxy)propyl]methylamine