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N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}piperidine-1-sulfonamide
ethyl 1-[3-(1,2-oxazinan-2-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
4-{[(1-hydroxycyclohexyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
(4aS,8aR)-1-(3-aminopropyl)-N-(furan-2-ylmethyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
(2S)-1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
2-[2-(4-chloro-3-methylphenoxy)-1-hydroxyethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
5-(3-cyclopropyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3R,4R)-1-[3-(1H-imidazol-1-yl)propyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-methyl-2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-{[2-(2-methylpropoxy)phenyl]methyl}acetamide
1-(2-fluorophenyl)-4-{[3-({1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl}piperazine
4-(5-acetylthiophene-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[2-(pyrrolidin-1-yl)ethyl]-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperazine-1-sulfonamide
1-[2-(3-methylthiophen-2-yl)ethyl]-2-(thiophen-3-yl)-1H-imidazole
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-hydroxy-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-4-(piperidin-1-ylmethyl)benzamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(5-fluoro-2-methylbenzenesulfonyl)piperidine
N-[3-(cyclohexylsulfanyl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenoxypropanamide
2-{2-[2-amino-3-cyano-6-(4-hydroxyphenyl)-5-methylpyridin-4-yl]phenoxy}acetic acid
(1-{[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}cyclopentyl)methanol
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
(3S,4S)-1-(6-methylpyridazin-3-yl)-4-(naphthalen-2-yl)piperidin-3-ol
4,4,4-trifluoro-1-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}butan-1-one
2-(2-{[(3-methyl-1-benzofuran-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-(oxan-4-ylmethyl)acetamide
6-(cyclobutylamino)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
(3S)-N-tert-butyl-2-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(2-hydroxyethyl)-8-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2-(thiophen-2-ylformamido)propanamide
3-methyl-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-[3-(oxolan-2-yl)propyl]urea
3-(2-phenoxyethyl)-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}piperidin-4-amine
1-[(2-aminopyridin-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(3S,4R)-1-(2,6-diaminopyrimidin-4-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-(2-ethoxyethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)benzonitrile
4-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1,2,5-tetramethyl-1H-pyrrole-3-carboxamide
N-{5-[(2R)-2-amino-2-cyclohexylacetamido]-2-methoxyphenyl}pentanamide
1-(6-carbamoyl-2H-1,3-benzodioxol-5-yl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxylic acid
1-{4-methyl-2-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]pyrimidin-5-yl}ethan-1-one
N-methyl-N-[2-(morpholin-4-yl)propyl]oxan-4-amine
N-{2-[(7-chloro-4-methylquinolin-2-yl)amino]ethyl}acetamide