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2-(1-methylpyrrolidin-3-yl)-9-[2-(thiophen-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,9aR)-8-[(2-chlorophenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-fluoro-3-methyl-2-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1H-indole
2-[1-(cyclopropylmethyl)-4-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl 2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
3-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N-(2-methylpropyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-ethyl-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-(6-aminopyridin-3-yl)-2-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]acetic acid
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[4-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}urea
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
4-{2-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
4-(cyclopropylsulfamoyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
[(5-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(1S,5R)-6-(3-chloro-5-methoxybenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-(4-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}-6-methylpyrimidin-2-yl)phenol
5-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(pyridin-4-yl)-N-[1-(thiophen-2-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aR,8aS)-1-(1H-indole-6-carbonyl)-6-(2-phenylethyl)-decahydro-1,6-naphthyridine
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(naphthalene-2-carbonyl)piperidine
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-4-methoxy-N,3,5-trimethylbenzamide
5-{[2-(phenylcarbamoyl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
methyl 4-{[(1-methyl-1H-1,2,3-triazol-4-yl)amino]methyl}benzoate
4-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-[4-(dimethylamino)phenyl]-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-5-methylthiophene-2-carboxamide
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-butylpiperidine-1-carboxamide
2-cyclopropyl-1-[2-(2,2-diphenylethyl)morpholin-4-yl]ethan-1-one
(1-{3-[(5,6-dimethylpyrimidin-4-yl)amino]propyl}piperidin-2-yl)methanol
2-({1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
6-fluoro-2-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
2-[4-(4-methoxypyrimidin-2-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
4-[3-(3-methoxypyrrolidine-1-carbonyl)benzenesulfonyl]-1-methylpiperazin-2-one
4'-(2,2-dimethylpropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(1H-indazol-6-yl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
2-[2-(dimethylamino)ethyl]-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-{3-[(cyclopropylamino)methyl]-6,7-dimethoxyquinolin-2-yl}piperidine-3-carboxylate
2-phenyl-N-[3-(piperidine-1-carbonyl)phenyl]pyrrolidine-1-carboxamide
{6-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]pyridin-2-yl}methanol
1-[(3-methylpyridin-2-yl)methyl]-6-[(1-phenylethyl)amino]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
(3-{2-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-(1H-indol-3-yl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
1-(2-aminoethyl)-N-cyclohexyl-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide