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6-[2-(4-fluorophenyl)morpholine-4-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
2-(3-methylphenyl)-4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
1-[2-(4-fluorobenzenesulfonyl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
7-(4-chlorophenyl)-2-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2-({2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-3-phenoxypropanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1H-pyrazol-1-yl)propanamide
(2S)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}propanamide
3-(aminomethyl)-4-[2-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-{[(adamantan-2-yl)amino]methyl}-5-(4-methylpiperazine-1-carbonyl)phenyl)acetamide
1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-[(2S)-2-amino-2-phenylacetyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(azepan-1-yl)-2-oxoethyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
N3-[3-(2-fluorophenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
7-fluoro-3-{[(3-hydroxypropyl)amino]methyl}-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
1-[1-(1-propylpiperidin-4-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(1S,3R)-3-amino-N-(3-phenylphenyl)cyclopentane-1-carboxamide
N-methyl-5-oxo-1-phenyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
7-(2-phenoxyethyl)-1,2-dihydroisoquinolin-1-one
4-[(4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}furan-2-yl)methyl]morpholine
4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-2-methoxyphenol
8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-hydroxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
7-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-5-(oxan-4-yl)-1H-1,2,4-triazole
3-{[3-(1H-imidazol-2-yl)propyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
4-(4,6-dimethylpyrimidin-2-yl)-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)piperazine-1-carboxamide
[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-[3-({4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)acetamide
3-(2,3-dimethylquinoxalin-6-yl)-1-methyl-1-(oxan-2-ylmethyl)urea
5-(3-phenylpiperazine-1-carbonyl)-2-(propan-2-yl)pyrimidine
1-[3-(methylsulfanyl)propyl]-4-(pyridin-3-yl)piperazine
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
(2S,4S)-4-[(adamantan-2-yl)amino]-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(1,3-dihydroxypropan-2-yl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-{[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]amino}acetate
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(thiophen-2-yl)ethyl]propanamide
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
2-[2-(butan-2-yl)phenoxy]-N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]acetamide
N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-N4,N4-dimethylpyrimidine-2,4-diamine
5-{1-[2-(ethanesulfonyl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyridin-2-amine
1-[2-(2-phenylethyl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
1-[1-(2-phenylethyl)-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
N-benzyl-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine