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4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methylbenzoyl)piperidine
N-{[1-(4-fluorophenyl)cyclopentyl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](thiophen-2-ylmethyl)amino}butan-1-ol
1-(2-{4-[(6-chloropyridin-3-yl)methyl]morpholin-2-yl}ethyl)-3-ethylurea
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,N-dimethyl-2-[(1S,5R)-3-[(6-methylpyridin-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(5-acetylthiophen-3-yl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]acetamide
ethyl 3-(2-methoxyethyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-3-carboxylate
3-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(1-methyl-2-oxopyrrolidin-3-yl)urea
5-{3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-5-methylpyrrolidin-2-one
(1R,5S)-3-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-acetyl-2,4-dimethyl-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-pyrrole-3-carboxamide
1-[2-methoxy-5-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-methyl-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine-2-carboxylic acid
2-[({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)amino]-1-phenylethan-1-ol
(1R,5R)-6-(cyclopropylmethyl)-N-[4-(methylsulfanyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1R,3S)-7-(3-hydroxypyridine-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-ethyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-4-(thiophen-2-yl)butan-1-one
5-[2-(4-fluorophenyl)morpholine-4-carbonyl]-N-phenylpyrimidin-2-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-(2,4,6-trimethyl-3-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazol-2-yl}phenyl)ethan-1-one
2,5-dimethyl-4-[3-(propan-2-yloxy)phenyl]pyrimidine
3-(furan-2-yl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-phenyl-3-{[2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl]formamido}propanamide
5-ethyl-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
4-methoxy-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
1-cyclohexyl-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-methyl-1H-1,2,4-triazole
2-(2-ethyl-1H-imidazol-1-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
4-(4-chlorophenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-(cyclopent-3-en-1-yl)-7-(4-methylbenzoyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(3-methyl-1H-indol-2-yl)methyl]amine
4-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
(2E)-3-(1,3-benzothiazol-2-yl)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]prop-2-enamide
2-(3-chlorophenoxy)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(1R,5S,6R)-N-{2-[ethyl(3-methylphenyl)amino]ethyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
(1S,4S)-2-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-5-methyl-2,5-diazabicyclo[2.2.1]heptane
2-(morpholin-3-yl)-N-(1-oxo-2,3,4,9-tetrahydro-1H-carbazol-7-yl)acetamide
2-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
N-(1-carbamoylcyclopentyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-(1-methoxypropan-2-yl)-15-methyl-13-oxo-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-(4-fluorophenyl)-N-(1,4-oxazepan-6-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-2-(2-methyl-1H-indol-3-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
(cyclohex-3-en-1-ylmethyl)({3-[(dimethylamino)methyl]phenyl}methyl)methylamine