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2-(methylamino)-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,4-diazepan-6-ol
8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[4-(1-ethyl-3-phenyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-1λ6-thiolane-1,1-dione
6-oxo-1-(3-phenylpropyl)piperidine-3-carboxylic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-hydroxypyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethoxy)ethan-1-ol
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
3-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
1-[2-(6-hydroxy-1,4-oxazepan-4-yl)-2-oxoethyl]-2-methyl-1H-indole-3-carbonitrile
1-({5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
2-(furan-2-yl)-N-[1-(4-methylpyridin-2-yl)propyl]-2-oxoacetamide
6-(2-aminoethyl)-N,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]pyrimidin-4-amine
1-(benzyloxy)-8-(3-phenoxypropanoyl)-1,8-diazaspiro[4.5]decan-2-one
2-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(thiophen-2-yl)-1,3-thiazole
(3aR,6aR)-2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-2-(pyridin-3-yl)-N-(2,2,2-trifluoroethyl)pyrimidine-5-carboxamide
N-(1-{1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[(6-methoxypyridin-3-yl)methyl]-1-methyl-2-phenylpiperazine
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methylphenyl)methyl]piperidine
2-(2-methyl-1H-imidazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
1-methyl-4-(1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)piperazine
2-tert-butyl-N-(4-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methoxyphenyl)methyl]acetamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[2-(thiophen-3-yl)acetyl]-decahydro-2,7-naphthyridine-2-sulfonamide
2-{5-[(3-chloro-5-fluorophenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(cyclopropylmethyl)pyrrolidin-2-one
(3S,4S)-1-(3-fluoro-2-methoxybenzoyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
methyl 2-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-4-(pyrimidin-5-yl)phenoxy}acetate
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-5-oxopyrrolidine-3-carboxamide
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2,4-dimethylpyrimidine
(4aR,7aS)-1-benzyl-4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-[(4-benzoylpiperazin-1-yl)methyl]-2-propylpyrimidine
8-methoxy-2-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
N,N-bis(prop-2-en-1-yl)-3-[(thiophen-2-ylmethyl)amino]benzamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1,2,4-oxadiazol-3-ylmethyl)piperidine
N,2,2-trimethyl-N-{[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}oxan-4-amine
5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
9-methyl-3-(2-propylpyridine-4-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclopentanecarbonylpiperidin-3-ol
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-2-sulfonamide
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one