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(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(2,5-dimethylfuran-3-carbonyl)piperidine
1-(2,4-dimethylphenoxy)-3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]propan-2-ol
2-[(1S,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
ethyl 1-ethyl-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-(propan-2-yl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
1-{[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
9-[(2-chloro-5-fluorophenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,2-dicyclopropyl-4-hydroxy-N-[(3-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide
1-[1-cyclohexyl-3-(2-methoxyphenoxymethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
3-[8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]propane-1,2-diol
methyl (2R)-2-(4-hydroxyphenyl)-2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}acetate
1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[(2-ethoxypyridin-3-yl)methyl]-4-phenylpyrimidine-5-carboxamide
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
6,6-dimethyl-1-(2-methylphenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
dimethyl(3-{2-[1-(4-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-{4-[(2,4-dimethyl-3-oxopiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
8-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S,4R)-4-[2-(2-hydroxyphenyl)acetamido]-1-(3-methylbut-2-en-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
4-ethyl-3-{1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[5-(3-methoxypiperidine-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
5-{[4-(3,4-dichlorophenyl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
4-({5-[(2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,4-oxazepane
6-methyl-2-(2-phenylethyl)-3-(piperidine-1-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-oxo-2-phenyl-N-[2-(piperidin-1-yl)ethyl]acetamide
6-chloro-2-[4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
1-{3-[4-(adamantan-1-yl)piperazin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(3-fluoro-4-phenylbenzoyl)piperidine
3-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2,8-diazaspiro[4.5]decane
N-(1,1-dioxo-1λ6-thiolan-3-yl)-5-methyl-N-(prop-2-en-1-yl)-1-propyl-1H-pyrazole-4-carboxamide
1-(6-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}pyridin-2-yl)ethan-1-ol
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}urea
5-[(2,3-difluoro-6-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
2-(dimethylamino)-8-[3-methoxy-2-(prop-2-yn-1-yloxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4,4,4-trifluoro-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
1,2-dimethyl-5-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
1-[3-methyl-1-(pyridin-3-yl)butyl]-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
(3S,9aR)-3-benzyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-({2-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(naphthalen-1-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[(2R)-1-hydroxybutan-2-yl]-1-[2-(propylsulfanyl)phenyl]urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1'-[(8-methoxyquinolin-2-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]