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3-(dimethyl-1,2-oxazol-4-yl)-1-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)urea
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
(4aS,8aR)-1-(3-aminopropyl)-6-[(2-methylpyrimidin-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-(2-methoxyethyl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenyl-N-(thian-4-yl)propanamide
[2-(1H-imidazol-1-yl)ethyl](methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-5-propyl-1,2-oxazole
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-cyclohexylpiperazine
(1S,4S)-2-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
5-chloro-4-methyl-6-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-amine
2-butyl-8-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[cyclohexyl(methyl)amino]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyridine-3-carboxamide
6,7-dimethoxy-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-oxopiperidin-1-yl)acetamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
6-chloro-3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
9-(3-fluoro-4-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}-1-[3-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
4-(cyclopropylmethyl)-1-[2-(2,4,6-trifluorophenyl)acetyl]-1,4-diazepan-5-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-{[4-(2-ethoxyethyl)piperazin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-methyl-8-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-2,8-diazaspiro[5.5]undecane
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}quinoxalin-2-amine
2-cyclopropyl-4-methyl-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]pyrimidine-5-carboxamide
N,N-dimethyl-2-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}phenyl)acetamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
1-{3-methyl-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
3-(2-hydroxyphenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazole-5-carboxamide
8-methoxy-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-cyclopentyl-2-methoxybenzamide
(3S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-phenylbutanamide
4-methylphenyl (7S,9aR)-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[(3S,4S)-4-methoxypyrrolidin-3-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-acetyl-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1H-pyrazole-5-carboxamide
2-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N3-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(4-methylphenyl)-3-(oxolan-3-ylformamido)propanamide
5-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,3,4-oxadiazol-2-amine
(3S,4S)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3R,4R)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-cyclohexyl-N3-(2-hydroxybutyl)-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
6-[(3R,5S)-3,5-bis(hydroxymethyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidin-3-yl]acetamide
4-{2-[(5-methyl-4-{1-[4-(propan-2-yloxy)benzoyl]piperidin-3-yl}pyrimidin-2-yl)sulfanyl]ethyl}morpholine
3-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-methoxybenzamide