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{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-{[(3-ethoxy-2-hydroxypropyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aS,8aR)-6-(5-acetylpyridin-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine-3-carboxylate
2-[1-(1H-pyrazole-4-carbonyl)azetidin-3-yl]-1H-1,3-benzodiazole
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
8-chloro-2-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)quinoline
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-methoxy-N-[3-({[2-(morpholin-4-yl)ethyl]carbamoyl}amino)phenyl]acetamide
(3S,4S)-4-cyclopropyl-1-[2-(pyrazin-2-yl)acetyl]pyrrolidine-3-carboxylic acid
3-(4-{1-[(3-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)prop-2-yn-1-ol
8-cyclopropanecarbonyl-2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-fluoro-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethylimidazo[1,2-a]pyridine-2-carboxamide
8-cyclopropanecarbonyl-2-(1-ethyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
(2S)-2-amino-1-(3,3-diphenylpiperidin-1-yl)-3-hydroxypropan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
(3aR,6aR)-2-acetyl-5-(quinolin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(5-chloro-2-propoxyphenyl)methyl]oxane-4-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-(1-methylpiperidin-2-yl)propanamide
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-[(1-propylcyclobutyl)methyl]acetamide
1-[(3S)-1-benzylpyrrolidin-3-yl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
3-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propan-1-ol
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-3-yl)benzoic acid
N-ethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
(3S,4S)-1-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
3-{[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-1-methyl-1H-indole
3-[2-(furan-2-yl)azepane-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-methylazepane-2-carboxamide
2-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-cyclohexyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(3-fluorophenyl)propan-1-one
6-({1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]hex-5-en-2-yl}oxy)-N,N-dimethylpyrazin-2-amine
methyl (2S,4S)-1-methyl-4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-amido)pyrrolidine-2-carboxylate
(2S,4S)-1-benzyl-N-ethyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
{4-[(4-chlorophenyl)methyl]-1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}methanol
2-[4-(2,5-dimethylphenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-4-methyl-1,3-oxazole-5-carboxamide
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(oxan-4-yl)piperazine
[(3S,5R)-1-(2,6-dimethylpyrimidine-4-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(4-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-4-yl)acetamide
5-[4-(aminomethyl)piperidin-1-yl]-2-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,3-dihydropyridazin-3-one