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1'-(1H-1,2,3-triazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]
N-[(5-methylthiophen-2-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-methyl-3-{N-methyl-1-[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}butanamide
4-[2-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)-1H-pyrrol-1-yl]benzonitrile
5-ethyl-1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(dimethylamino)-7-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinolin-6-ylmethyl)pyrrolidin-3-yl]methanol
3-(4-methyl-1,3-thiazol-5-yl)-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}propanamide
1-(4-fluorophenyl)-4-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)piperazine
3-ethyl-4-({4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-2-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(1H-pyrazol-1-yl)butanamide
6-ethyl-2-methyl-4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}quinoline
(3S,4R)-1-(3-chlorothiophene-2-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
[1-(2-chloro-4-fluorobenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(2S,4R)-4-(dimethylamino)-1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxylic acid
N-ethyl-5-[4-(2-methylphenyl)piperazine-1-carbonyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
3-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]imidazolidine-2,4-dione
1-{2-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]ethyl}pyrrolidin-2-one
1-[(3-fluorophenyl)methyl]-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazine
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-4-phenyl-N-(pyridin-2-ylmethyl)benzamide
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
1'-[(5-acetylthiophen-3-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(methanesulfonylmethyl)piperidine
N-[3-(1H-indol-2-yl)phenyl]-1-propylpiperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
(3aS,6aS)-2-methyl-5-(5-phenoxyfuran-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(cyclohexylmethyl)-N-methyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine-4-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(furan-3-ylmethyl)-N-methylacetamide
7-propyl-2-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(piperidin-1-ylmethyl)piperidine
6-{1-[3-methyl-4-(morpholin-4-yl)benzoyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
1-(cyclohexylmethyl)-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
N-[(3R,4R)-3-hydroxy-1-(5,6,7,8-tetrahydroquinolin-2-yl)piperidin-4-yl]pyrazine-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
(4aS,7aR)-N-[(4-methoxyphenyl)methyl]-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-[1'-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(4aR,7aS)-1-acetyl-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-chlorophenyl)-4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-(3-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propyl)-1H-pyrazole
1-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
N-[(3R,4R)-3-hydroxy-1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(naphthalen-1-yl)ethyl]propanamide
1-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole